IP Library Granted Patent US 8,389,543
Granted Patent B2
US 8,389,543 · App. 13/293,891 · Granted Mar 5, 2013

Metalloenzyme inhibitor compounds

Inventors: William J. Hoekstra (Durham, NC); Robert J. Schotzinger (Raleigh, NC); Stephen W. Rafferty (Durham, NC)
Assignee: Viamet Pharmaceuticals, Inc.
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Quick Facts
Patent No.
US 8,389,543
App. No.
13/293,891
Granted
Mar 5, 2013
Kind
B2
Abstract

The instant invention describes compounds having metalloenzyme modulating activity, and methods of treating diseases, disorders or symptoms thereof mediated by such metalloenzymes.

Claims (9)

1. A compound of formula (III) or salt thereof:

wherein X is CH, Y is CH, R 2 is alkyl, R 3 is OH, and R 4 and R 5 are independently H, halogen, alkoxy, fluoroalkoxy containing 1-5 fluorines, cyano, carboxamido, optionally substituted aryl, or optionally substituted heteroaryl.

2. The compound of claim 1 that is:

1-(6,7-Dimethoxynaphthalen-2-yl)-2-methyl-1-(1H-1,2,3-triazol-4-yl)propan-1-ol (1);

1-(6,7-Bis(difluoromethoxy)naphthalen-2-yl)-2-methyl-1-(1H-1,2,3-triazol-4-yl)propan-1-ol (3);

2-Methyl-1-(6-(oxazol-5-yl)naphthalen-2-yl)-1-(1H-1,2,3-triazol-4-yl)propan-1-ol (4);

2-methyl-1-(1H-1,2,3-triazol-4-yl)-1-(6-(2,2,2-trifluoroethoxy)naphthalen-2-yl )propan-1-ol (12);

1-(6-(difluoromethoxy)naphthalen-2-yl)-2-methyl-1-(1H-1,2,3-triazol-4-yl)propan-1-ol (13);

or salt thereof.

Assignments (4)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Mar 18, 2021
From: INNOCRIN PHARMACEUTICALS HOLDINGS, LLC
To: KEMBI THERAPEUTICS PTY LTD
Reel/Frame 055635/0883 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Mar 8, 2021
From: INNOCRIN PHARMACEUTICALS, INC.
To: INNOCRIN PHARMACEUTICALS HOLDINGS, LLC
Reel/Frame 055518/0691 →
CHANGE OF NAME Recorded Oct 27, 2014
From: VIAMET PHARMACEUTICALS, INC.
To: INNOCRIN PHARMACEUTICALS, INC.
Reel/Frame 034066/0202 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Feb 2, 2012
From: HOEKSTRA, WILLIAM J.; SCHOTZINGER, ROBERT J.; RAFFERTY, STEPHEN W.
To: VIAMET PHARMACEUTICALS, INC.
Reel/Frame 027639/0689 →
Continuity (2)
Provisional Application 61413395 · Nov 13, 2010
Related Publication 20120129886A1 · May 24, 2012