IP Library Granted Patent US 8,426,468
Granted Patent B2
US 8,426,468 · App. 13/445,679 · Granted Apr 23, 2013

Use of medium chain triglycerides for the treatment and prevention of alzheimer'S disease and other diseases resulting from reduced neuronal metabolism

Inventor: Samuel T. Henderson (Golden, CO)
Assignee: Accera, Inc.
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Quick Facts
Patent No.
US 8,426,468
App. No.
13/445,679
Granted
Apr 23, 2013
Kind
B2
Abstract

Methods and compositions for treating or preventing, the occurrence of senile dementia of the Alzheimer's type, or other conditions arising from reduced neuronal metabolism and leading to lessened cognitive function are described. In a preferred embodiment the administration of triglycerides or fatty acids with chain lengths between 5 and 12, to said patient at a level to produce an improvement in cognitive ability.

Claims (15)

1. A method of treating loss of cognitive function caused by reduced neuronal metabolism, wherein said treatment comprises oral administration of a dosage unit of medium chain triglyceride to a patient such that the blood level of D-beta-hydroxybutyrate in the patient is raised to about 1-10 mM or patient urinary excretion of D-beta-hydroxybutyrate is in the range 5 mg/dL to 160 mg/dL causing hyperketonemia in the patient, wherein the patient has a diet wherein carbohydrate intake is not restricted, resulting in ketone bodies being utilized for energy in the brain.

2. The method of claim 1 , wherein said administration is in a single dose.

3. The method of claim 1 , wherein said loss of cognitive function is caused by Alzheimer's Disease or Mild Cognitive Impairment.

4. The method claim 1 , wherein said medium chain triglyceride is administered at a dose of about 0.5 g/kg/day to about 10 g/kg/day.

5. The method of claim 1 , further comprising coadministering L-carnitine.

6. The method of claim 5 , wherein said administration is oral, and said medium chain triglyceride is administered at a dose of about 0.5 g/kg/day to about 10 g/kg/day and said L-carnitine is administered at a dose of about 0.5 mg/kg/day to about 10 mg/kg/day.

7. The method of claim 1 , wherein said medium chain triglyceride is emulsified.

8. The method of claim 7 , further comprising coadministering L-carnitine.

9. The method of claim 8 , wherein said emulsified medium chain triglyceride and L-carnitine or a derivative of L-carnitine are administered in a formulation comprising 10-500 g emulsified medium chain triglyceride and 10-2000 mg L-carnitine.

10. A method of treating loss of cognitive function caused by reduced neuronal metabolism, wherein said treatment comprises oral administration of 10 g to 50 g of medium chain triglyceride to a patient over the course of one day such that the blood level of D-beta-hydroxybutyrate in the patient is raised to about 1-10 mM or patient urinary excretion of D-beta-hydroxybutyrate is in the range 5 mg/dL to 160 mg/dL causing hyperketonemia in the patient, wherein the patient has a diet wherein carbohydrate intake is not restricted, resulting in ketone bodies being utilized for energy in the brain.

11. The method of claim 10 , wherein said administration is in a single dose.

12. The method of claim 10 , wherein said loss of cognitive function is caused by Alzheimer's Disease or Mild Cognitive Impairment.

13. The method of claim 10 , further comprising coadministering L-carnitine.

14. The method of claim 10 , wherein said medium chain triglyceride is emulsified.

15. The method of claim 14 , further comprising coadministering L-carnitine.

Assignments (4)
RELEASE OF SECURITY INTEREST Recorded Feb 10, 2025
From: NESTLÉ HEALTH SCIENCE US HOLDINGS, INC.
To: CERECIN INC.
Reel/Frame 070168/0946 →
CHANGE OF NAME Recorded Aug 26, 2020
From: ACCERA, INC.
To: CERECIN INC.
Reel/Frame 053605/0604 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Sep 5, 2012
From: HENDERSON, SAMUEL T.
To: ACCERA, INC.
Reel/Frame 028902/0153 →
PATENT SECURITY AGREEMENT Recorded Jul 24, 2012
From: ACCERA, INC.
To: NESTLE HEALTH SCIENCE US HOLDINGS, INC., AS COLLATERAL AGENT
Reel/Frame 028624/0001 →
Continuity (4)
Continuation 11331673 · Jan 13, 2006
Continuation 09845741 · May 1, 2001
Provisional Application 60200980 · May 1, 2000
Related Publication 20120196932A1 · Aug 2, 2012