IP Library Granted Patent US 8,932,588
Granted Patent B2
US 8,932,588 · App. 13/508,207 · Granted Jan 13, 2015

Treatment of cancer involving mutated KRAS or BRAF genes

Inventors: Norbert A. Kienzle (Dundas Valley, AU); Anthony G. Doyle (Drummoyne, AU); Tony Rowe (Sandringham, AU)
Assignee: Teva Pharmaceuticals Australia Pty. Ltd.
C07K16/30A61K2039/505C07K2316/95C07K2317/24C07K2317/41C07K2317/732
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Quick Facts
Patent No.
US 8,932,588
App. No.
13/508,207
Granted
Jan 13, 2015
Kind
B2
Abstract

The present invention provides a method of treating cancer in a subject wherein the cancer comprises mutated KRAS or BRAF genes. The method comprises administering to the subject an effective amount of an antibody or antigen binding fragment thereof wherein the antibody or antigen binding fragment thereof competes with SC104 for binding to the human colon cancer cell line Colo205.

Claims (12)

1. A method of treating cancer in a subject wherein the cancer comprises mutated KRAS or BRAF genes, the method comprising administering to the subject an effective amount of an antibody or antigen binding fragment thereof comprising a light chain and heavy chain amino acid sequence combination selected from the group consisting of SEQ ID NO:7/SEQ ID NO:25, SEQ ID NO:7/SEQ ID NO:50, SEQ ID NO:7/SEQ ID NO:94, SEQ ID NO:8/SEQ ID NO:26 and SEQ ID NO:8/SEQ ID NO:38.

2. A method of treating cancer in a subject, the method comprising testing the cancer for the presence of mutated KRAS or BRAF genes and, if the cancer has a mutated KRAS or a mutated BRAF gene, administering to the subject an effective amount of an antibody or antigen binding fragment thereof comprising a light chain and heavy chain amino acid sequence combination selected from the group consisting of SEQ ID NO:7/SEQ ID NO:25, SEQ ID NO:7/SEQ ID NO:50, SEQ ID NO:7/SEQ ID NO:94, SEQ ID NO:8/SEQ ID NO:26 and SEQ ID NO:8/SEQ ID NO:38.

3. A method as claimed in claim 1 , wherein the cancer is selected from the group consisting of colon cancer, pancreatic cancer, and gastric cancer.

4. A method as claimed in claim 1 , wherein the antibody is a deimmunized.

5. A method as claimed in claim 1 , wherein the antibody or antigen binding fragment comprises SEQ ID NO:7 and SEQ ID NO:94.

6. The method as claimed in claim 1 , wherein the antibody or antigen binding fragment thereof has been glyco-engineered to enhance antibody-dependent cell-mediated cytotoxicity.

7. A method as claimed in claim 2 , wherein the cancer is selected from the group consisting of colon cancer, pancreatic cancer, and gastric cancer.

8. A method as claimed in claim 2 , wherein the antibody is a deimmunized.

9. A method as claimed in claim 2 , wherein the antibody or antigen binding fragment comprises SEQ ID NO:7 and SEQ ID NO:94.

10. The method as claimed in claim 2 , wherein the antibody or antigen binding fragment thereof has been glyco-engineered to enhance antibody-dependent cell-mediated cytotoxicity.

11. The method as claimed in claim 1 , wherein the antibody or antigen binding fragment thereof competes with SC104 for binding to the human colon cancer cell line Colo205.

12. The method as claimed in claim 2 , wherein the antibody or antigen binding fragment thereof competes with SC104 for binding to the human colon cancer cell line Colo205.

Assignments (2)
CHANGE OF NAME Recorded Nov 13, 2013
From: CEPHALON AUSTRALIA PTY LTD.
To: TEVA PHARMACEUTICALS AUSTRALIA PTY. LTD.
Reel/Frame 031590/0470 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jul 19, 2012
From: KIENZLE, NORBERT A.; DOYLE, ANTHONY G.; ROWE, TONY
To: CEPHALON AUSTRALIA PTY. LTD.
Reel/Frame 028584/0561 →
Priority Claims (1)
AU 2010904107 · Sep 13, 2010 · national
Continuity (2)
Provisional Application 61258518 · Nov 5, 2009
Related Publication 20120244151A1 · Sep 27, 2012