IP Library Granted Patent US 9,284,347
Granted Patent B2
US 9,284,347 · App. 13/522,030 · Granted Mar 15, 2016

Chromatographic method for purifying FC-containing proteins

Inventors: Christian Eckermann (Biberach an der Riss, DE); Dorothee Ambrosius (Laupheim, DE); Franz Nothelfer (Biberach an der Riss, DE); Thomas Rathjen (Biberach an der Riss, DE)
Assignee: Boehringer Ingelheim International GmbH
C07K1/22A61K39/39591C07K16/00C07K2317/14
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Quick Facts
Patent No.
US 9,284,347
App. No.
13/522,030
Granted
Mar 15, 2016
Kind
B2
Abstract

The present invention relates to methods of depleting impurities, in particular host cell proteins (HCP) and DNA from cell culture supernatants by means of protein A chromatography using a novel washing buffer.

Claims (26)

1. A method of depleting impurities from a composition that contains a protein which comprises the Fc domain of an immunoglobulin (target protein), by protein-A chromatography, comprising the steps of:

a. applying a mobile phase which contains the target protein to a stationary phase which contains protein A, under conditions in which the target protein binds to the stationary phase;

b. applying a washing buffer with a pH of between 4 and 8 as mobile phase, containing

i. arginine in a concentration of 0.1-1 mol/l,

ii. sodium chloride in a concentration of 0.2 to 2 mol/l,

iii. an alcohol selected from among isopropanol, n-propanol and ethanol, in a concentration of 5-30% (w/v) and

iv. polyvinylpyrrolidone in a concentration of 0.05-2% (w/v);

c. using an elution buffer as mobile phase under conditions in which the target protein is eluted from the stationary phase.

2. The method according to claim 1 , wherein the arginine concentration in the washing buffer is 0.4-0.6 mol/l.

3. The method according to claim 1 , wherein the sodium chloride concentration in the washing buffer is 0.9-1.1 mol/l.

4. The method according to claim 1 , wherein the alcohol in the washing buffer is isopropanol in a concentration of 10-20% (w/v).

5. The method according to claim 1 , wherein polyvinylpyrrolidone (PVP) is in a concentration of 0.1-2% (w/v).

6. The method according to claim 1 , wherein the impurities are host cell proteins (HCP).

7. A method of depleting impurities from a composition that contains a protein which comprises the Fc domain of an immunoglobulin (target protein), by protein-A chromatography, comprising the steps of:

a. applying a mobile phase which contains the target protein to a stationary phase which contains protein A, under conditions in which the target protein binds to the stationary phase;

b. applying a washing buffer with a pH of between 5 and 8 as mobile phase, containing

i. arginine in a concentration of 0.1—1 mol/l,

ii. sodium chloride in a concentration of 0.2 to 2 mol/l,

iii. an alcohol selected from among isopropanol, n-propanol and ethanol, in a concentration of 5—30% (w/v) and

iv. polyvinylpyrrolidone in a concentration of 0.05—2% (w/v);

c. using an elution buffer as mobile phase under conditions in which the target protein is eluted from the stationary phase.

8. The method according to claim 7 , wherein the arginine concentration in the washing buffer is 0.4—0.6 mol/l.

9. The method according to claim 7 , wherein the sodium chloride concentration in the washing buffer is 0.9—1.1 mol/l.

10. The method according to claim 7 , wherein the alcohol in the washing buffer is isopropanol in a concentration of 10—20% (w/v).

11. The method according to claim 7 , wherein polyvinylpyrrolidone (PVP) is in a concentration of 0.1—2% (w/v).

12. The method according to claim 7 , wherein the impurities are host cell proteins (HCP).

Assignments (1)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded May 7, 2015
From: ECKERMANN, CHRISTIAN; AMBROSIUS, DOROTHEE; NOTHELFER, FRANZ; RATHJEN, THOMAS
To: BOEHRINGER INGELHEIM INTERNATIONAL GMBH
Reel/Frame 035583/0696 →
Priority Claims (2)
EP 10151416 · Jan 22, 2010 · regional
EP 10171975 · Aug 5, 2010 · regional
Continuity (1)
Related Publication 20130197197A1 · Aug 1, 2013