IP Library Granted Patent US 8,507,460
Granted Patent B2
US 8,507,460 · App. 13/650,739 · Granted Aug 13, 2013

Substituted 3′,5′-cyclic phosphates of purine nucleotide compounds and pharmaceutical compositions for the treatment of viral infections

Inventors: Dominique Surleraux (Wauthier-Braine, BE); Cyril B. Dousson (Canet, FR); Christophe Claude Parsy (Jacou, FR)
Assignee: Idenix Pharmaceuticals, Inc.
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Quick Facts
Patent No.
US 8,507,460
App. No.
13/650,739
Granted
Aug 13, 2013
Kind
B2
Abstract

Provided herein are compounds, compositions and methods for the treatment of Flaviviridae infections, including HCV infections. In certain embodiments, compounds and compositions of nucleoside derivatives are disclosed, which can be administered either alone or in combination with other anti-viral agents.

Claims (26)

1. A compound of Formula I:

or a pharmaceutically acceptable salt, solvate, stereoisomeric form, tautomeric form or polymorphic form thereof, wherein

R 1 is lower alkyl or hydrogen, and

R 2 is lower alkyl.

2. The compound of claim 1 wherein R 1 is hydrogen, methyl, ethyl, n-propyl, isopropyl, n-butyl, isobutyl or t-butyl.

3. The compound of claim 1 wherein R 2 is methyl, ethyl, n-propyl, isopropyl, n-butyl, isobutyl, 2-butyl, cyclopentyl, cyclobutyl, cyclopropyl or t-butyl.

4. The compound of claim 1 according to formula Ia or Ib:

or a pharmaceutically acceptable salt, solvate, stereoisomeric form, tautomeric form or polymorphic form thereof.

5. The compound of claim 1 according to formula II:

or a pharmaceutically acceptable salt, solvate, stereoisomeric form, tautomeric form or polymorphic form thereof.

6. The compound of claim 1 according to formula IIa or IIb:

or a pharmaceutically acceptable salt, solvate, stereoisomeric form, tautomeric form or polymorphic form thereof.

7. A pharmaceutical composition comprising the compound of claim 1 and a pharmaceutically acceptable excipient, carrier or diluent.

8. The pharmaceutical composition of claim 7 , wherein the composition is an oral formulation.

9. A pharmaceutical composition comprising the compound of claim 5 and a pharmaceutically acceptable excipient, carrier or diluent.

10. The pharmaceutical composition of claim 9 , wherein the composition is an oral formulation.

11. A method for the treatment of a host infected with a hepatitis C virus, comprising the administration of an effective treatment amount of a compound of claim 1 .

12. The method of claim 11 , wherein the host is a human.

13. The method of claim 11 , wherein said administration directs a substantial amount of said compound or pharmaceutically acceptable salt or stereoisomer thereof to the liver of said host.

14. The method of claim 11 , wherein said compound is administered in combination or alternation with a second anti-viral agent optionally selected from the group consisting of an interferon, a ribavirin, an interleukin, a NS3 protease inhibitor, a cysteine protease inhibitor, a phenanthrenequinone, a thiazolidine derivative, a thiazolidine, a benzanilide, a helicase inhibitor, a polymerase inhibitor, a nucleotide analogue, a gliotoxin, a cerulenin, an antisense phosphorothioate oligodeoxynucleotide, an inhibitor of IRES-dependent translation, and a ribozyme.

15. The method of claim 14 , wherein the second agent is selected from the group consisting of telaprevir, bocepravir, pegylated interferon alpha 2a, interferon alphacon-1, natural interferon, albuferon, interferon beta-1a, omega interferon, interferon alpha, interferon gamma, interferon tau, interferon delta and interferon γ-1b.

16. A method for the treatment of a host infected with a hepatitis C virus, comprising the administration of an effective treatment amount of a compound of claim 5 .

17. The method of claim 16 , wherein the host is a human.

18. The method of claim 16 , wherein said administration directs a substantial amount of said compound or pharmaceutically acceptable salt or stereoisomer thereof to the liver of said host.

19. The method of claim 16 , wherein said compound is administered in combination or alternation with a second anti-viral agent optionally selected from the group consisting of an interferon, a ribavirin, an interleukin, a NS3 protease inhibitor, a cysteine protease inhibitor, a phenanthrenequinone, a thiazolidine derivative, a thiazolidine, a benzanilide, a helicase inhibitor, a polymerase inhibitor, a nucleotide analogue, a gliotoxin, a cerulenin, an antisense phosphorothioate oligodeoxynucleotide, an inhibitor of IRES-dependent translation, and a ribozyme.

20. The method of claim 19 , wherein the second agent is selected from the group consisting of telaprevir, bocepravir, pegylated interferon alpha 2a, interferon alphacon-1, natural interferon, albuferon, interferon beta-1a, omega interferon, interferon alpha, interferon gamma, interferon tau, interferon delta and interferon γ-1b.

Assignments (2)
CHANGE OF NAME Recorded Jul 30, 2015
From: IDENIX PHARMACEUTICALS, INC.
To: IDENIX PHARMACEUTICALS LLC
Reel/Frame 036234/0158 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Dec 5, 2012
From: SURLERAUX, DOMINIQUE; DOUSSON, CYRIL B.; PARSY, CHRISTOPHE CLAUDE
To: IDENIX PHARMACEUTICALS, INC.
Reel/Frame 029409/0946 →
Continuity (4)
Provisional Application 61547625 · Oct 14, 2011
Provisional Application 61555329 · Nov 3, 2011
Provisional Application 61703084 · Sep 19, 2012
Related Publication 20130095064A1 · Apr 18, 2013