IP Library Granted Patent US 9,114,133
Granted Patent B2
US 9,114,133 · App. 13/658,943 · Granted Aug 25, 2015

Method of improving diastolic dysfunction

Inventor: Samuel C. Dudley, Jr. (Chicago, IL)
Assignees: U.S. DEPT. OF VETERANS AFFAIRS; THE BOARD OF TRUSTEES OF THE UNIV. OF ILLINOIS
A61K31/40A61K31/519A61K38/44
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Quick Facts
Patent No.
US 9,114,133
App. No.
13/658,943
Granted
Aug 25, 2015
Kind
B2
Abstract

A method of treating, preventing, reversing, or ameliorating diastolic dysfunction includes reducing S-glutathionylated myosin binding protein-C (MyBP-C) level by administering to a host in need thereof a therapeutically effective amount of tetrahydrobiopterin (BH 4 ).

Claims (14)

1. A method of treating, reversing, or ameliorating diastolic dysfunction in a host with normal systolic function, comprising:

a) providing a host with normal systolic function with an ejection fraction of 50% or greater, and in need of treating, reversing, or ameliorating diastolic dysfunction; and

b) reducing S-glutathionylated myosin binding protein-C (MyBP-C) level by administering to the host a therapeutically effective amount of tetrahydrobiopterin (BH 4 ).

2. The method of claim 1 , wherein the step of administering comprises:

administering BH 4 in at least one form selected from the group consisting of a dietary supplement, a composition, a pharmaceutical composition, and a combination thereof.

3. The method of claim 1 , wherein the step of administering comprises:

administering BH 4 orally.

4. The method of claim 1 , wherein the host is a human.

5. The method of claim 1 , wherein the host is an animal.

6. A method of treating, preventing, reversing, or ameliorating diastolic dysfunction, comprising: modulating post-translational modification of myosin binding protein-C (MyBP-C) level by administering to a host in need thereof a therapeutically effective amount of tetrahydrobiopterin (BH4).

7. The method of claim 6 , wherein the step of administering comprises: administering BH4 in at least one form selected from the group consisting of a dietary supplement, a composition, a pharmaceutical composition, and a combination thereof.

8. The method of claim 6 , wherein the step of administering comprises: administering BH4 orally.

9. The method of claim 6 , wherein the host is a human.

10. The method of claim 6 , wherein the host is an animal.

Assignments (2)
CONFIRMATORY LICENSE Recorded Aug 20, 2013
From: THE BOARD OF TRUSTEES OF THE UNIVERSITY OF ILLINOIS ON BEHALF OF ITS OFFICE OF TECHNOLOGY MANAGEMENT OFFICE AT THE UNIVERSITY OF ILLINOIS AT CHICAGO
To: NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT
Reel/Frame 031041/0115 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Feb 13, 2013
From: DUDLEY, SAMUEL C. JR.
To: U. S. DEPARTMENT OF VETERANS AFFAIRS; BOARD OF TRUSTEES OF THE UNIVERSITY OF ILLINOIS, THE
Reel/Frame 029928/0157 →
Continuity (4)
Continuation In Part 11895883 · Aug 27, 2007
Provisional Application 60840368 · Aug 25, 2006
Provisional Application 61552500 · Oct 28, 2011
Related Publication 20130065903A1 · Mar 14, 2013