IP Library Granted Patent US 9,426,995
Granted Patent B2
US 9,426,995 · App. 13/763,087 · Granted Aug 30, 2016

Compositions and methods for controlling nematodes

Inventors: Urszula Slomczynska (Ballwin, MO); Matt W. Dimmic (Maryland Heights, MO); Al Wideman (St. Louis, MO); William P. Haakenson, Jr. (St. Louis, MO)
Assignee: Monsanto Technology LLC
A01N43/82C07D413/04C07D413/06
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Quick Facts
Patent No.
US 9,426,995
App. No.
13/763,087
Granted
Aug 30, 2016
Kind
B2
Abstract

Compositions and processes for controlling nematodes are described herein, e.g., nematodes that infest plants or animals. The compounds include oxazoles, oxadiazoles and thiadiazoles.

Claims (43)

1. A coated seed wherein the coating comprises a compound of Formula VII or a salt thereof,

wherein,

A is aryl, arylalkyl, aryloxo, arylthio, heteroaryl, heteroarylalkyl, heteroaryloxo, or heteroarylthio, each of which may be optionally independently substituted with one or more substituents selected from the group consisting of halo, C 1 -C 6 haloalkyl, C 6 -C 10 aryl, C 4 -C 7 cycloalkyl, C 2 -C 6 alkyl, C 2 -C 6 alkenyl, C 2 -C 6 alkynyl, C 6 -C 10 aryl(C 1 -C 6 )alkyl, C 6 -C 10 aryl(C 2 -C 6 )alkenyl, C 6 -C 10 aryl(C 2 -C 6 ) alkynyl, C 1 -C 6 hydroxyalkyl, amino, ureido, cyano, C 1 -C 6 acylamino, hydroxy, thiol, C 1 -C 6 acyloxy, azido, OCH 3 , OCF 3 , and C(H)O;

and

C is pyrrolyl, pyrrolyloxo, pyrrolythio, or pyrrolylalkyl, each of which may be optionally independently substituted with one or more substituents selected from the group consisting of CH 3 , C 2 -C 10 alkyl, cycloalkyl, heterocycle, hydroxyalkyl, and halogen.

2. The coated seed of claim 1 comprising a compound of formula VIIa or a salt thereof,

wherein,

R 1 and R 5 are independently selected from the group consisting of hydrogen, CH 3 , F, Cl, Br, CF 3 and OCF 3 ;

R 2 and R 4 are independently selected from the group consisting of hydrogen, F, Cl, Br, and CF 3 ;

R 3 is selected from the group consisting of hydrogen, CH 3 , CF 3 , F, Cl, Br, OCF 3 , OCH 3 , CN, and C(H)O;

R 6 , R 7 , R g and R 9 are independently selected from the group consisting of hydrogen, CH 3 , C 2 -C 10 alkyl, cycloalkyl, heterocycle, and halogen; and

X is a bond, CH 2 , O, or S.

3. The coated seed of claim 1 wherein the coating is applied to the seed as a composition comprising the compound in an aqueous carrier.

4. The coated seed of claim 3 wherein the composition comprises a surfactant.

5. The coated seed of claim 3 wherein the composition comprises a co-solvent.

6. The seed of claim 3 wherein the coating further comprises a pesticide.

7. The composition coated seed of claim 6 wherein the pesticide is selected from the group consisting of avermectin, ivermectin, milbemycin, imidacloprid, aldicarb, oxamyl, fenamiphos, fosthiazate, metam sodium, etridiazole, penta-chloro-nitrobenzene (PCNB), flutolanil, metalaxyl, mefenoxam, fosetyl-al, silthiofam, fludioxonil, myclobutanil, azoxystrobin, chlorothalonil, propiconazole, tebuconazole, pyraclostrobin, trifloxysulfuron, glyphosate and halosulfuron.

8. A coated seed wherein the coating comprises a compound of Formula XII or a salt thereof,

wherein,

A is arylor arylalkyl, each of which may be optionally independently substituted with one or more substituents selected from the group consisting of halo, C 1 -C 6 haloalkyl, C 6 -C 10 aryl, C 4 -C 7 cycloalkyl, C 2 -C 6 alkyl, C 2 -C 6 alkenyl, C 2 -C 6 alkynyl, C 6 -C 10 aryl(C 1 -C 6 )alkyl, C 6 -C 10 aryl(C 2 -C 6 )alkenyl, C 6 -C 10 aryl(C 2 -C 6 ) alkynyl, C 1 -C 6 hydroxyalkyl, amino, ureido, cyano, C 1 -C 6 acylamino, hydroxy, thiol, C 1 -C 6 acyloxy, azido, C 1 -C 6 alkoxy and carboxy, and C(H)O; and

C is selected from the group consisting of thienyl, furanyl, oxazolyl, and isoxazolyl, each of which can be optionally independently substituted with one or more substituents selected from the group consisting of fluorine, chlorine, CH 3 , and OCF 3 ; and

X is CH 2 , O,or S.

9. The coated seed of claim 8 comprising a compound of Formula XIIa or a salt thereof,

wherein,

R 1 and R 5 are independently selected from the group consisting of hydrogen, CH 3 , F, Cl, Br, CF 3 , and OCF 3 ;

R 2 and R 4 are independently selected from the group consisting of hydrogen, F, Cl, Br, and CF 3 ;

R 3 is selected from the group consisting of hydrogen, CH 3 , CF 3 , F, Cl, Br, OCF 3 , OCH 3 , CN, and C(H)O;

R 7 , R g and R 9 are independently selected from the group consisting of hydrogen, F, Cl, CH 3 , and OCF 3 ;

E is O, or S; and

X is CH 2 , O, or S.

10. The coated seed of claim 8 comprising a compound of Formula XIIb or a salt thereof,

wherein,

R 1 and R 5 are independently selected from the group consisting of hydrogen, CH 3 , F, Cl, Br, CF 3 , and OCF 3 ;

R 2 and R 4 are independently selected from the group consisting of hydrogen, F, Cl, Br, and CF 3 ;

R 3 is selected from the group consisting of hydrogen, CH 3 , CF 3 , F, Cl, Br, OCF 3 , OCH 3 , CN, and C(H)O;

R 6 , R g and R 9 are independently selected from the group consisting of hydrogen, F, Cl, CH 3 , and OCF 3 ;

E is O, or S; and

X is CH 2 , O, or S.

11. The coated seed of claim 8 wherein the coating is applied to the seed as a composition comprising the compound in an aqueous carrier.

12. The coated seed of claim 11 wherein the composition comprises a surfactant.

13. The coated seed of claim 11 wherein the composition comprises a co-solvent.

14. The coated seed of claim 11 wherein the coating further comprises a pesticide.

15. The coated seed of claim 14 wherein the pesticide is selected from the group consisting of avermectin, ivermectin, milbemycin, imidacloprid, aldicarb, oxamyl, fenamiphos, fosthiazate, metam sodium, etridiazole, penta-chloro-nitrobenzene (PCNB), flutolanil, metalaxyl, mefenoxam, fosetyl-al, silthiofam, fludioxonil, myclobutanil, azoxystrobin, chlorothalonil, propiconazole, tebuconazole, pyraclostrobin, trifloxysulfuron, glyphosate and halosulfuron.

Assignments (4)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jul 3, 2013
From: WIDEMAN, AL
To: DIVERGENCE, INC.
Reel/Frame 030737/0251 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jun 3, 2013
From: SLOMCZYNSKA, URSZULA; DIMMIC, MATT W.; HAAKENSON, WILLIAM P., JR.
To: DIVERGENCE INC.
Reel/Frame 030533/0649 →
MERGER Recorded Jun 3, 2013
From: DIVERGENCE, INC.
To: MONSANTO COMPANY
Reel/Frame 030533/0736 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jun 3, 2013
From: MONSANTO COMPANY
To: MONSANTO TECHNOLOGY LLC
Reel/Frame 030533/0751 →
Continuity (4)
Continuation 12904724 · Oct 14, 2010
Continuation 12703750 · Feb 10, 2010
Provisional Application 61151482 · Feb 10, 2009
Related Publication 20130217570A1 · Aug 22, 2013