IP Library Granted Patent US 8,753,638
Granted Patent B2
US 8,753,638 · App. 13/766,659 · Granted Jun 17, 2014

Compositions and methods comprising histidyl-TRNA synthetase splice variants having non-canonical biological activities

Inventors: Jie Zhou (Kowloon, HK); Ching-Fun Lau (New Territories, HK); Zhiwen Xu (Kowloon, HK); Wing-Sze Lo (Chai Wan, HK); Kristi Helen Piehl (San Diego, CA); Leslie Ann Greene (San Diego, CA)
Assignee: aTyr Pharma, Inc.
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Quick Facts
Patent No.
US 8,753,638
App. No.
13/766,659
Granted
Jun 17, 2014
Kind
B2
Abstract

Isolated histidyl-tRNA synthetase splice variant polynucleotides and polypeptides having non-canonical biological activities are provided, as well as compositions and methods related thereto.

Claims (26)

1. A method for treating an inflammatory or autoimmune condition in a subject in need thereof, comprising administering to the subject a pharmaceutical composition that comprises a pharmaceutically acceptable carrier and a histidyl-tRNA synthetase (HRS) polypeptide splice variant, where the HRS polypeptide is about 50-175 amino acids in length and comprises 50 or more contiguous amino acids of SEQ ID NO:6 or a variant thereof having at least 95% sequence identity to SEQ ID NO:6, and where the HRS polypeptide comprises a WHEP domain and lacks a functional aminoacylation domain.

2. The method of claim 1 , where the HRS polypeptide is about 50-70 amino acids in length.

3. The method of claim 2 , where the HRS polypeptide comprises the amino acid sequence of SEQ ID NO:6 or a variant thereof having at least 95% sequence identity to SEQ ID NO:6.

4. The method of claim 3 , where the HRS polypeptide consists essentially of SEQ ID NO:6.

5. The method of claim 1 , where the HRS polypeptide is about 175 amino acids in length.

6. The method of claim 5 , where the HRS polypeptide comprises the amino acid sequence of SEQ ID NO:9 or a variant thereof having at least 95% sequence identity to SEQ ID NO:9.

7. The method of claim 6 , where the HRS polypeptide comprises the amino acid sequence of SEQ ID NO:9.

8. The method of claim 7 , where the HRS polypeptide consists essentially of SEQ ID NO:9.

9. A method for treating an inflammatory or autoimmune condition in a subject in need thereof, comprising administering to the subject a pharmaceutical composition that comprises a pharmaceutically acceptable carrier and a histidyl-tRNA synthetase (HRS) polypeptide, where the HRS polypeptide is about 212 amino acids in length and comprises 50 or more contiguous amino acids of SEQ ID NO:11 or a variant thereof having at least 95% sequence identity to SEQ ID NO:11, and where the HRS polypeptide comprises a WHEP domain and lacks a functional aminoacylation domain.

10. An isolated histidyl-tRNA synthetase (HRS) splice variant polypeptide, for use in a method of reducing inflammatory activity wherein the HRS polypeptide comprises the amino acid sequence of SEQ ID NO: 11, or a variant thereof having at least 95% sequence identity to SEQ ID NO: 11, where the HRS polypeptide comprises a WHEP domain and lacks a functional aminoacylation domain.

11. The method of claim 10 , where the HRS polypeptide comprises the amino acid sequence of SEQ ID NO:11.

12. The method of claim 11 , where the HRS polypeptide consists essentially of SEQ ID NO:11.

13. A method for treating an inflammatory or autoimmune condition in a subject in need thereof, comprising administering to the subject a pharmaceutical composition that comprises a pharmaceutically acceptable carrier and a histidyl-tRNA synthetase (HRS) polypeptide, where the HRS polypeptide is about 40-80 amino acids in length and comprises about 40 or more contiguous amino acids of SEQ ID NO:6 or a variant thereof having at least 95% sequence identity to SEQ ID NO:6 where the HRS polypeptide comprises a WHEP domain.

14. The method of claim 13 , where the HRS polypeptide comprises about 50 or more amino acids of SEQ ID NO:6.

15. The method of claim 13 , where the HRS polypeptide consists essentially of SEQ ID NO:6.

16. A method for treating an inflammatory or autoimmune condition in a subject in need thereof, comprising administering to the subject a pharmaceutical composition that comprises a pharmaceutically acceptable carrier and a histidyl-tRNA synthetase (HRS) polypeptide, where the HRS polypeptide consists essentially of a WHEP domain from human histidyl-tRNA synthetase (HRS).

17. The method of any of claim 1 , 9 , 13 , or 16 , where the HRS polypeptide is modified by pegylation.

18. The method of any of claim 1 , 9 , 13 , or 16 , where the HRS polypeptide further comprises a heterologous fusion partner.

19. The method of claim 18 , where the heterologous fusion partner comprises an Fc fragment.

20. The method of any of claim 1 , 9 , 13 , or 16 , where the HRS polypeptide is a recombinant polypeptide.

21. The method of any of claim 1 , 9 , 13 , or 16 , where the HRS polypeptide is a synthetic polypeptide.

22. The method of any of claim 1 , 9 , 13 , or 16 , where the HRS polypeptide comprises at least one chemical or enzymatic derivation at one or more constituent amino acids where the at least one chemical or enzymatic derivation is selected from acetylation, hydroxylation, methylation, amidation, glycosylation, and lipidation.

23. The method of any of claim 1 , 9 , 13 , or 16 , where the pharmaceutical composition is formulated with histidine.

24. The method of any of claim 1 , 9 , 13 , or 16 , where the pharmaceutical composition comprises a surfactant.

25. The method of any of claim 1 , 9 , 13 , or 16 , where the pharmaceutical composition is administered by oral, parenteral, intravenous, intranasal, inhalation, aerosol, intracranial, or intramuscular administration.

26. An isolated recombinant histidyl-tRNA synthetase (HRS) polypeptide, for use in a method of reducing inflammatory activity wherein the HRS polypeptide is 50-175 amino acids in length and comprises at least 50 contiguous amino acids of SEQ ID NO: 6, or a variant thereof having at least 95% sequence identity to SEQ ID NO: 6, where the HRS polypeptide comprises a WHEP domain and lacks a functional aminoacylation domain.

Assignments (4)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Oct 3, 2014
From: ZHOU, JIE; LAU, CHING FUN; XU, ZHIWEN; LO, WING SZE; PIEHL, KRISTI HELEN; GREENE, LESLIE ANN
To: ATYR PHARMA, INC.
Reel/Frame 033884/0598 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Oct 3, 2014
From: ZHOU, JIE; LAU, CHING FUN; XU, ZHIWEN; LO, WING-SZE
To: PANGU BIOPHARMA LIMITED
Reel/Frame 033884/0612 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Oct 3, 2014
From: PANGU BIOPHARMA LIMITED
To: ATYR PHARMA, INC.
Reel/Frame 033884/0639 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Oct 3, 2014
From: ATYR PHARMA, INC.
To: PANGU BIOPHARMA LIMITED
Reel/Frame 033889/0988 →
Continuity (4)
Continuation 12725272 · Mar 16, 2010
Provisional Application 61239747 · Sep 3, 2009
Provisional Application 61160630 · Mar 16, 2009
Related Publication 20130243766A1 · Sep 19, 2013