IP Library Granted Patent US 9,868,728
Granted Patent B2
US 9,868,728 · App. 13/876,869 · Granted Jan 16, 2018

Quinazoline derivatives, compositions, and uses related thereto

Inventors: John David Lambeth (Decatur, GA); Thota Ganesh (Alpharetta, GA); Susan M. Smith (Acworth, GA); Aiming Sun (Atlanta, GA)
Assignee: Emory University
C07D417/12A01N1/0226A61K8/4953A61K31/517A61K31/519A61K45/06A61Q19/08
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Quick Facts
Patent No.
US 9,868,728
App. No.
13/876,869
Granted
Jan 16, 2018
Kind
B2
Abstract

The invention relates to quinazoline derivatives, compositions, and methods related thereto. In certain embodiments, the invention relates to inhibitors of NADPH-oxidase.

Claims (4)

1. A pharmaceutical formulation comprising 6-chloro-3-(3-(dimethylamino)propyl)-2-thioxo-2,3-dihydroquinazolin-4(1H)-one or salt thereof and a pharmaceutically acceptable carrier.

2. The pharmaceutical formulation of claim 1 in the form of a tablet, soft or hard gelatin or non-gelatin capsule, or caplet.

3. The pharmaceutical formulation of claim 1 wherein the pharmaceutically acceptable carrier is selected from dicalcium phosphate dihydrate, calcium sulfate, sucrose, glucose, dextrose, lactose, sorbitol, dextrose, cellulose, starch, gelatin, silicone dioxide, titanium oxide, magnesium aluminum silicate, magnesium stearate, calcium stearate, stearic acid, glycerol behenate, polyethylene glycol, talc, mineral oil, and an acrylic polymer.

4. The pharmaceutical formulation of claim 1 wherein the pharmaceutically acceptable carrier is a lubricant, surfactant, or enteric coating.

Assignments (1)
CONFIRMATORY LICENSE Recorded Apr 15, 2013
From: EMORY UNIVERSITY
To: NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT
Reel/Frame 030211/0825 →
Continuity (2)
Provisional Application 61407925 · Oct 29, 2010
Related Publication 20130225612A1 · Aug 29, 2013