IP Library Granted Patent US 9,181,216
Granted Patent B2
US 9,181,216 · App. 14/083,205 · Granted Nov 10, 2015

4′-O-substituted isoindoline derivatives and compositions comprising and methods of using the same

Inventors: Alexander L. Ruchelman (Cream Ridge, NJ); George W. Muller (Rancho Santa Fe, CA); Hon-Wah Man (Princeton, NJ); Roger Shen-Chu Chen (Edison, NJ)
Assignee: Celgene Corporation
C07D401/04A61K31/454A61K31/4709A61K45/06C07D401/14C07D405/14C07D409/14
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Quick Facts
Patent No.
US 9,181,216
App. No.
14/083,205
Granted
Nov 10, 2015
Kind
B2
Abstract

Provided are 4′-O substituted isoindoline compounds, and pharmaceutically acceptable salts, solvates, clathrates, stereoisomers, and prodrugs thereof. Methods of use, and pharmaceutical compositions of these compounds are disclosed.

Claims (8)

1. A compound of formula:

or a pharmaceutically acceptable salt or stereoisomer thereof, wherein:

Y is C═O or CH 2 ; and

R 1 is alkyl substituted with one or more groups selected from alkoxy, halo, carboxy, alkylaminocarbonyl, alkoxycarbonyl, nitro, nitrile, haloalkyl, hydroxy, and alkylsulfonyl.

2. The compound of claim 1 , wherein Y is C═O.

3. The compound of claim 1 , wherein Y is CH 2 .

4. The compound of claim 1 , wherein the compound is:

5. A pharmaceutical composition comprising a compound of claim 1 , or a pharmaceutically acceptable salt, or stereoisomer thereof.

Assignments (2)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Dec 18, 2017
From: CHEN, ROGER SHEN-CHU
To: CELGENE CORPORATION
Reel/Frame 044425/0995 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Oct 2, 2015
From: RUCHELMAN, ALEXANDER L.; MULLER, GEORGE W.; MAN, HON-WAH
To: CELGENE CORPORATION
Reel/Frame 036746/0387 →
Continuity (4)
Division 13410216 · Mar 1, 2012
Continuation 12077715 · Mar 19, 2008
Provisional Application 60919323 · Mar 20, 2007
Related Publication 20140073669A1 · Mar 13, 2014