IP Library Granted Patent US 9,248,163
Granted Patent B2
US 9,248,163 · App. 14/094,042 · Granted Feb 2, 2016

Insulin-like growth factor binding protein 7 for treatment of cancer

Inventors: Michael Green (Boylston, MS); Narendra Wajapeyee (Hamden, MA)
Assignee: University of Massachusetts
A61K38/1754C12Q1/6886G01N33/5743
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Quick Facts
Patent No.
US 9,248,163
App. No.
14/094,042
Granted
Feb 2, 2016
Kind
B2
Abstract

Methods of treating a tumor in a subject include identifying a subject having, at risk for, or suspected of having a tumor, and administering to the subject an effective amount of an IGFBP7 agent if the tumor has increased Ras-BRAF-MEK-Erk signaling, is dependent for growth and/or survival upon the Ras-BRAF-MEK-Erk signaling pathway, and/or expresses an activated or oncogenic BRAF or RAS.

Claims (26)

1. A method of treating a tumor in a subject, the method comprising:

identifying a subject having a tumor that has a cell having increased Ras-BRAF-MEK-Erk signaling, is dependent for growth and/or survival upon the Ras-BRAF-MEK-Erk signaling pathway, and/or expresses an activated or oncogenic BRAF or RAS; and

administering to the subject an effective amount of an IGFBP7 polypeptide at least 80% identical to SEQ ID NO:1 or SEQ ID NO:7, thereby treating the tumor.

2. The method of claim 1 , wherein the tumor is a cancer.

3. The method of claim 2 , wherein the cancer is a melanoma.

4. The method of claim 2 , wherein the cancer is a carcinoma, breast cancer, ovarian cancer, pancreatic cancer, colon cancer, colorectal carcinoma, or papillary thyroid carcinoma.

5. The method of claim 2 , wherein the cancer expresses an activated or oncogenic BRAF or RAS.

6. The method of claim 2 , wherein the activated or oncogenic BRAF is BRAFV600E.

7. The method of claim 1 , wherein the oncogenic BRAF is BRAFV600E.

8. The method of claim 1 , wherein the polypeptide is at least 85% identical to SEQ ID NO:1 or SEQ ID NO:7.

9. The method of claim 1 , wherein the polypeptide is conjugated to a heterologous moiety.

10. The method of claim 9 , wherein the heterologous moiety is a heterologous polypeptide sequence.

11. The method of claim 1 , wherein the IGFBP7 agent consists of a polypeptide at least 80% identical to SEQ ID NO:1 or SEQ ID NO:7.

12. The method of claim 11 , wherein the polypeptide is at least 85% identical to SEQ ID NO:1 or SEQ ID NO:7.

13. The method of claim 1 , wherein the IGFBP7 polypeptide is administered by introducing to the subject a nucleic acid encoding a polypeptide at least 85% identical to SEQ ID NO:1 or SEQ ID NO:7.

14. The method of claim 13 , wherein the nucleic acid is in a viral vector.

15. The method of claim 14 , wherein the viral vector is an adenovirus, adeno-associated virus, retrovirus, or lentivirus vector.

16. The method of claim 1 , wherein the IGFBP7 agent is administered topically, systemically, or locally.

17. The method of claim 16 , wherein the IGFBP7 agent is administered locally by a drug-releasing implant.

18. A method of inhibiting proliferation of a cell that has increased Ras-BRAF-MEK-Erk signaling, is dependent for growth and/or survival upon the Ras-BRAF-MEK-Erk signaling pathway, and/or expresses an activated or oncogenic BRAF or RAS, the method comprising

identifying a cell that has increased Ras-BRAF-MEK-Erk signaling, is dependent for growth and/or survival upon the Ras-BRAF-MEK-Erk signaling pathway, and/or expresses an activated or oncogenic BRAF or RAS; and

administering to the cell an effective amount of an IGFBP7 polypeptide.

19. The method of claim 18 , wherein the cell is a tumor cell.

20. A method of treating a melanoma in a subject, the method comprising:

identifying a subject having, at risk for, or suspected of having a melanoma; and

administering to the subject an effective amount of an IGFBP7 polypeptide at least 80% identical to SEQ ID NO:1 or SEQ ID NO:7, thereby treating the melanoma.

Assignments (2)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Feb 13, 2014
From: GREEN, MICHAEL; WAJAPEYEE, NARENDRA
To: UNIVERSITY OF MASSACHUSETTS
Reel/Frame 032211/0355 →
CONFIRMATORY LICENSE Recorded Dec 16, 2013
From: UNIVERSITY OF MASSACHUSETTS MEDICAL SCHOOL
To: NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT
Reel/Frame 031817/0625 →
Continuity (5)
Continuation 13269091 · Oct 7, 2011
Continuation 12209028 · Sep 11, 2008
Provisional Application 60993211 · Sep 11, 2007
Provisional Application 61092230 · Aug 27, 2008
Related Publication 20140178339A1 · Jun 26, 2014