IP Library Granted Patent US 9,248,150
Granted Patent B2
US 9,248,150 · App. 14/094,864 · Granted Feb 2, 2016

Use of transplatin to prevent hearing loss

Inventors: Vickram Ramkumar (Springfield, IL); Debashree Mukherjea (Springfield, IL); Len Rybak (Springfield, IL)
Assignee: The Board of Trustees of the Southern Illinois University
A61K33/24A61K9/0019A61K9/0046A61K45/06
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Quick Facts
Patent No.
US 9,248,150
App. No.
14/094,864
Granted
Feb 2, 2016
Kind
B2
Abstract

Methods and compositions for treating and preventing toxic side effects of platinum-based chemotherapy agents are disclosed, in which transplatin is administered to a subject. Transplatin is shown to have protective effects against cisplatin-induced ototoxicity, nephotoxicity and neurotoxicity. Anti-inflammatory activity of transplatin is demonstrated and methods and compositions for treating and preventing inflammatory pain are described.

Claims (19)

1. A method of treating or preventing ototoxic effects of an ototoxic agent in a subject in need thereof, the method comprising administering to the subject a therapeutically effective amount of transplatin.

2. The method of claim 1 , wherein the method comprises administering the transplatin to the subject before exposure of the subject to the ototoxic agent.

3. The method of claim 1 , wherein the method comprises administering the transplatin to the subject during exposure of the subject to the ototoxic agent.

4. The method of claim 1 , wherein the method comprises administering the transplatin to the subject after exposure of the subject to the ototoxic agent.

5. The method of claim 1 , wherein the transplatin is administered via intraperitoneal injection or trans-tympanic injection.

6. The method of claim 1 , wherein the transplatin is administered via oral administration.

7. The method of claim 1 , wherein the ototoxic agent is selected from a platinum-based chemotherapy agent, radiation, Meniere's disease, noise, and an aminoglycoside.

8. The method of claim 7 , wherein the ototoxic agent is noise.

9. The method of claim 7 , wherein the ototoxic agent is an aminoglycoside.

10. The method of claim 7 , wherein the ototoxic agent is a platinum-based chemotherapy agent.

11. The method of claim 2 , wherein the ototoxic agent is selected from a platinum-based chemotherapy agent, radiation, Meniere's disease, noise, and an aminoglycoside.

12. The method of claim 3 , wherein the ototoxic agent is selected from a platinum-based chemotherapy agent, radiation, Meniere's disease, noise, and an aminoglycoside.

13. The method of claim 4 , wherein the ototoxic agent is selected from a platinum-based chemotherapy agent, radiation, Meniere's disease, noise, and an aminoglycoside.

14. The method of claim 1 , wherein the amount of transplatin is between about 0.1 mg/kg and about 50 mg/kg.

15. The method of claim 1 , wherein the ototoxic agent is another therapeutic agent and the transplatin is administered simultaneously with the other therapeutic agent.

16. The method of claim 1 , wherein the ototoxic agent is another therapeutic agent and the transplatin is administered within about 24 hours before administration of the other therapeutic agent.

17. The method of claim 1 , wherein the ototoxic agent is another therapeutic agent and the transplatin is administered within about 24 hours after administration of the other therapeutic agent.

18. The method of claim 16 , wherein the ototoxic agent is another therapeutic agent and the transplatin is administered within about 1 to about 6 hours before administration of the other therapeutic agent.

19. The method of claim 17 , wherein the ototoxic agent is another therapeutic agent and the transplatin is administered within about 1 to about 6 hours after administration of the other therapeutic agent.

Assignments (2)
CONFIRMATORY LICENSE Recorded Feb 23, 2016
From: BOARD OF TRUSTEES OF SOUTHERN ILLINOIS UNIVERSITY
To: NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT
Reel/Frame 037894/0220 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Dec 17, 2013
From: RAMKUMAR, VICKRAM; MUKHERJEA, DEBASHREE; RYBAK, LEN
To: THE BOARD OF TRUSTEES OF THE SOUTHERN ILLINOIS UNIVERSITY
Reel/Frame 031801/0607 →
Continuity (3)
Division 12836398 · Jul 14, 2010
Provisional Application 61225772 · Jul 15, 2009
Related Publication 20140087006A1 · Mar 27, 2014