IP Library Granted Patent US 9,468,687
Granted Patent B2
US 9,468,687 · App. 14/147,674 · Granted Oct 18, 2016

Immuno gene therapy for treatment of cancer and hyperproliferative diseases

Inventors: Jason G. Fewell (Madison, AL); Majed Matar (Madison, AL); Jennifer Rice (Grant, AL); Danny H. Lewis (Hartselle, AL); Khursheed Anwer (Madison, AL)
Assignee: CLSN LABORATORIES, INC.
A61K47/34A61K9/0019A61K9/0085A61K31/17A61K31/28A61K31/337A61K31/4745A61K31/664A61K31/704A61K31/7068A61K31/7072A61K31/7076A61K33/24A61K38/208A61K39/39558A61K47/10A61K47/48969A61K48/005A61K48/0041B82Y5/00C12N15/87
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Quick Facts
Patent No.
US 9,468,687
App. No.
14/147,674
Granted
Oct 18, 2016
Kind
B2
Abstract

Pharmaceutical compositions comprising a nucleic acid, a gene delivery polymer, and at least one adjunctive chemotherapeutic drug for the treatment of mammalian cancer or hyperproliferative disorders and methods of using thereof for the treatment of mammalian cancer or hyperproliferative disorders by intratumoral, intraperitoneal or systemic injection.

Claims (13)

1. A therapy for the treatment of a solid primary or metastasized tumor in a subject, wherein the tumor is disseminated to the peritoneal cavity and is an ovarian tumor, pancreatic tumor, liver tumor, colorectal tumor, mesothelioma, or combinations thereof, comprising: administering a pharmaceutical composition to the subject, wherein the pharmaceutical composition comprises a DNA plasmid that encodes interleukin-12 and a lipopolymer, said lipopolymer including a polyethylenimine backbone wherein cholesterol and polyethylene glycol are each covalently linked to the polyethylenimine backbone; wherein the administering is intratumoral or intraperitoneal and wherein expression of interleukin-12 results in inhibition of tumors.

2. The therapy of claim 1 , wherein the therapy provides a systemic effect.

3. A method of delivering an anti-tumor molecule into a peritoneal cavity of a subject with a hyperproliferative disorder comprising: contacting cells in the peritoneal cavity with a pharmaceutical composition comprising (1) a DNA plasmid that encodes interleukin-12 and (2) a lipopolymer, wherein the lipopolymer comprises a polyethylenimine backbone, wherein cholesterol and polyethylene glycol are each covalently linked to the polyethylenimine backbone; wherein the delivering is intratumoral or intraperitoneal and wherein the interleukin-12 is expressed in the cells in the peritoneal cavity resulting in a decrease of the hyperproliferative cells.

4. The method of claim 3 , wherein the hyperproliferative disorder is ovarian tumor cells that have metastasized to the peritoneal cavity.

5. The method of claim 3 , wherein the hyperproliferative disorder is colorectal tumor cells that have metastasized to the peritoneal cavity.

6. The method of claim 3 , wherein the hyperproliferative disorder is pancreatic tumor cells that have metastasized to the peritoneal cavity.

7. The method of claim 3 , wherein the hyperproliferative disorder is liver tumor cells that have metastasized to the peritoneal cavity.

8. The method of claim 3 , wherein the hyperproliferative disorder is mesothelioma tumor cells that have metastasized to the peritoneal cavity.

9. A combination therapy for the treatment of a glioma tumor in a subject, comprising: administering a pharmaceutical composition to the subject, wherein the administering is intracranial and the pharmaceutical composition comprises a DNA plasmid that encodes interleukin-12 and a lipopolymer, said lipopolymer including a polyethylenimine backbone wherein cholesterol and polyethylene glycol are each covalently linked to the polyethylenimine backbone, such that interleukin-12 is expressed; and administering at least one chemotherapeutic or anticancer agent to the subject wherein said combination therapy results in inhibition of the glioma tumor.

10. The combination therapy of claim 9 , wherein the anticancer agent is an anti-cancer antibody or other immunotherapy.

11. The combination therapy of claim 9 , wherein the anticancer agent is selected from the group consisting of carmustine, gemcitabine, cyclophosphamide, cisplatin, and paclitaxel.

12. A therapy for the treatment of a glioma tumor in a subject, comprising: administering a pharmaceutical composition to the subject, wherein the pharmaceutical composition comprises a DNA plasmid that encodes interleukin-12 and a lipopolymer, said lipopolymer including a polyethylenimine backbone wherein cholesterol and polyethylene glycol are each covalently linked to the polyethylenimine backbone; wherein the administering is intracranial and wherein expression of interleukin-12 results in inhibition the glioma tumor.

13. A method of delivering an anti-tumor molecule into the brain of a subject with a hyperproliferative disorder comprising: contacting cells in the brain of the subject with a pharmaceutical composition comprising (1) a DNA plasmid that encodes interleukin-12 and (2) a lipopolymer, wherein the lipopolymer comprises a polyethylenimine backbone, wherein cholesterol and polyethylene glycol are each covalently linked to the polyethylenimine backbone; wherein the delivering is intracranial and wherein the interleukin-12 is expressed in the cells in the brain resulting in a decrease of the hyperproliferative cells.

Assignments (3)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Sep 22, 2014
From: EGEN, INC.
To: CLSN LABORATORIES, INC.
Reel/Frame 033788/0539 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jan 30, 2014
From: FEWELL, JASON; MATAR, MAJED; RICE, JENNIFER; LEWIS, DANNY; ANWER, KHURSHEED
To: EXPRESSION GENETICS, INC.
Reel/Frame 032094/0247 →
CHANGE OF NAME Recorded Jan 30, 2014
From: EXPRESSION GENETICS, INC.
To: EGEN, INC.
Reel/Frame 032141/0151 →
Continuity (4)
Continuation 13109473 · May 17, 2011
Continuation 11261931 · Oct 28, 2005
Provisional Application 60635042 · Dec 9, 2004
Related Publication 20140186375A1 · Jul 3, 2014