IP Library Granted Patent US 9,139,583
Granted Patent B2
US 9,139,583 · App. 14/169,775 · Granted Sep 22, 2015

Selective HDAC3 inhibitors

Inventors: John H. van Duzer (Georgetown, MA); Ralph Mazitschek (Belmont, MA)
Assignee: ACETYLON PHARMACEUTICALS, INC.
C07D471/04C07D209/34C07D215/54C07D231/56C07D235/06
View Patent ↗
Loading inventors, assignments & file history…
Monitor This Case
Get email alerts when status or documents change.
Order Certified Copies
Most orders are placed with the USPTO same day — all within 24 business hours.
Order via The Patent Place →
Pre-filled with this patent's details
Quick Facts
Patent No.
US 9,139,583
App. No.
14/169,775
Granted
Sep 22, 2015
Kind
B2
Abstract

Provided herein are inhibitors of HDAC3, as well as methods of treatment comprising administering those compounds to a subject in need thereof.

Claims (15)

1. A compound selected from the following:

or a pharmaceutically acceptable salt thereof.

2. A pharmaceutical composition comprising a compound of claim 1 , or a pharmaceutically acceptable salt thereof, together with a pharmaceutically acceptable carrier.

3. A method of treating type 2 diabetes, Huntington's disease, spinal and bulbar muscular atrophy, or lung cancer in a subject comprising administering to the subject a compound of claim 1 or a pharmaceutically acceptable salt thereof.

4. The method of claim 3 , wherein the disease is type 2 diabetes.

5. The method of claim 3 , wherein the disease is Huntington's disease.

6. The method of claim 3 , wherein the disease is spinal and bulbar muscular atrophy.

7. The method of claim 3 wherein the disease is lung cancer.

8. The method of claim 3 , wherein the subject is human.

9. A compound which is:

or a pharmaceutically acceptable salt thereof.

10. A compound which is:

or a pharmaceutically acceptable salt thereof.

11. A compound which is:

or a pharmaceutically acceptable salt thereof.

Assignments (2)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Nov 3, 2017
From: ACETYLON PHARMACEUTICALS INC
To: REGENACY PHARMACEUTICALS, LLC
Reel/Frame 044032/0220 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jun 25, 2014
From: VAN DUZER, JOHN H.; MAZITSCHEK, RALPH
To: ACETYLON PHARMACEUTICALS, INC.
Reel/Frame 033173/0923 →
Continuity (2)
Provisional Application 61759732 · Feb 1, 2013
Related Publication 20140249148A1 · Sep 4, 2014