IP Library Granted Patent US 9,314,452
Granted Patent B2
US 9,314,452 · App. 14/188,061 · Granted Apr 19, 2016

Treatment of amyotrophic lateral sclerosis (ALS) with ibudilast

Inventors: Michael E. Kalafer (San Diego, CA); Kenneth W. Locke (Carlsbad, CA); Kazuko Matsuda (Beverly Hills, CA); Richard E. Gammans (Edmond, OK)
Assignee: MediciNova, Inc.
A61K31/437
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Quick Facts
Patent No.
US 9,314,452
App. No.
14/188,061
Granted
Apr 19, 2016
Kind
B2
Abstract

Compositions and methods for treating progressive neurodegenerative diseases, and their associated symptoms by administration of ibudilast (3-isobutyryl-2-isopropylpyrazolo[1,5-a]pyridine).

Claims (12)

1. A method of treating a patient diagnosed with amyotrophic lateral sclerosis (ALS) comprising administering to said patient a therapeutically effective amount of ibudilast or a pharmaceutically acceptable salt thereof ranging between 1-240 mg/day.

2. The method of claim 1 in which the ibudilast or pharmaceutically acceptable salt thereof is administered for at least six months.

3. The method of claim 1 in which the ibudilast or pharmaceutically acceptable salt thereof is administered for at least one year.

4. The method of claim 1 in which the ibudilast or pharmaceutically acceptable salt thereof is administered for at least two years.

5. The method of claim 1 in which the ibudilast or pharmaceutically acceptable salt thereof is administered at least once daily.

6. The method of claim 1 in which the ibudilast or pharmaceutically acceptable salt thereof is administered orally.

7. The method of claim 1 in which the ibudilast or pharmaceutically acceptable salt thereof is administered in an amount of 30 mg to 240 mg daily.

8. The method of claim 1 in which the ibudilast or pharmaceutically acceptable salt thereof is administered in an amount of 30 mg to 120 mg daily.

9. The method of claim 1 in which the ibudilast or pharmaceutically acceptable salt thereof is administered in an amount of 1 mg to 120 mg daily.

10. The method of claim 1 in which the ibudilast or pharmaceutically acceptable salt thereof is administered in a total daily dosage amount selected from the group consisting of 30 mg/day, 60 mg/day, 90 mg/day and 120 mg/day.

11. A method of treating a patient diagnosed with amyotrophic lateral sclerosis (ALS) comprising administering to said patient a therapeutically effective amount of ibudilast or a pharmaceutically acceptable salt thereof ranging between about 0.1 and 200 mg/day.

12. The method of claim 11 in which the ibudilast or pharmaceutically acceptable salt thereof is administered in a total daily dosage amount selected from the group consisting of 30 mg/day, 60 mg/day, 90 mg/day and 120 mg/day.

Continuity (6)
Continuation 13725627 · Dec 21, 2012
Continuation 13402702 · Feb 22, 2012
Continuation 12169042 · Jul 8, 2008
Provisional Application 60929745 · Jul 11, 2007
Provisional Application 61042181 · Apr 3, 2008
Related Publication 20140171463A1 · Jun 19, 2014