IP Library Granted Patent US 9,745,631
Granted Patent B2
US 9,745,631 · App. 14/367,341 · Granted Aug 29, 2017

Methods for diagnosing and treating oncogenic kras-associated cancer

Inventors: Ronald A. DePinho (Houston, TX); Lewis Cantley (Cambridge, MA); Alec C. Kimmelman (Weston, MA); Haoqiang Ying (Houston, TX); Costas A. Lyssiotis (Boston, MA)
Assignees: Dana-Farber Cancer Institute, Inc.; Beth Israel Deaconess Medical Center, Inc.
C12Q1/6886A61K31/436A61K31/4412C12Q2600/112C12Q2600/118C12Q2600/158
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Quick Facts
Patent No.
US 9,745,631
App. No.
14/367,341
Granted
Aug 29, 2017
Kind
B2
Abstract

Methods for diagnosing and treating cancer associated with an oncogenic Kras mutation in a subject are provided.

Claims (17)

1. A method for treating a subject having a cancer comprising an oncogenic Kras mutation, the method comprising

detecting that a sample obtained from the subject comprises an elevated level of expression of ribulose-5-phosphate-3-epimerase (RPE) compared to a control sample lacking an oncogenic Kras mutation, and

inhibiting RPE or ribose 5-phosphate isomerase A (RPIA) in the subject, thereby treating the subject.

2. The method of claim 1 , wherein said subject has been previously determined or is simultaneously determined to have a cancer comprising the oncogenic Kras mutation.

3. The method of claim 2 , wherein said Kras mutation is selected from the group consisting of Kras G12D , Kras G12V , Kras G13D , Kras G12C , Kras Q61R Kras Q61L , Kras Q61K , Kras G12R , and Kras G12C .

4. The method of claim 1 , wherein said cancer is selected from the group consisting of pancreatic cancer, non-small cell lung cancer, colorectal cancer, and biliary cancer.

5. A method comprising:

(1) providing a sample from a subject, wherein the sample comprises an oncogenic Kras mutation;

(2) detecting that said sample comprises an elevated level of expression of ribulose-5-phosphate-3-epimerase (RPE) compared to a control sample lacking the oncogenic Kras mutation, and

(3) inhibiting RPE or ribose 5-phosphate isomerase A (RPIA) in the subject.

6. The method of claim 5 , wherein said subject has been previously determined or is simultaneously determined to comprise an oncogenic Kras mutation.

7. The method of claim 6 , wherein said Kras mutation is selected from the group consisting of Kras G12D , Kras G12V , Kras G13D , Kras G12C , Kras Q61R , Kras Q61L , Kras Q61K , Kras G12R , and Kras G12C .

8. The method of claim 5 , wherein the subject has pancreatic cancer, non-small cell lung cancer, colorectal cancer, or biliary cancer.

9. The method of claim 1 , wherein RPE is inhibited by administering to the subject an antisense oligonucleotide that targets RPE or a small interfering RNA that targets RPE.

10. The method of claim 1 , wherein RPIA is inhibited by administering to the subject an antisense oligonucleotide that targets RPIA or a small interfering RNA that targets RPIA.

11. The method of claim 5 , wherein RPE is inhibited by administering to the subject an antisense oligonucleotide that targets RPE or a small interfering RNA that targets RPE.

12. The method of claim 5 , wherein RPIA is inhibited by administering to the subject an antisense oligonucleotide that targets RPIA or a small interfering RNA that targets RPIA.

Assignments (3)
CONFIRMATORY LICENSE Recorded Jul 19, 2016
From: DANA-FARBER CANCER INST
To: NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT
Reel/Frame 039389/0470 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Dec 10, 2014
From: DEPINHO, RONALD A.; KIMMELMAN, ALEC C.; YING, HAOQIANG
To: DANA-FARBER CANCER INSTITUTE, INC.
Reel/Frame 034453/0552 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Dec 10, 2014
From: CANTLEY, LEWIS; LYSSIOTIS, COSTAS A.
To: BETH ISRAEL DEACONESS MEDICAL CENTER, INC.
Reel/Frame 034453/0663 →
Continuity (2)
Provisional Application 61578116 · Dec 20, 2011
Related Publication 20150126580A1 · May 7, 2015