IP Library Granted Patent US 9,365,542
Granted Patent B2
US 9,365,542 · App. 14/438,584 · Granted Jun 14, 2016

Modulators of resistant androgen receptor

Inventors: Minna D. Balbas (San Francisco, NY); Michael J. Evans (Pacifica, NY); Charles L. Sawyers (New York, NY); Yang Shen (Chicago, IL); David Hosfield (Chicago, IL); Geoffrey L. Greene (Chicago, IL)
Assignee: Memorial Sloan-Kettering Cancer Center
C07D401/04C07D233/86C07D235/02
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Quick Facts
Patent No.
US 9,365,542
App. No.
14/438,584
Granted
Jun 14, 2016
Kind
B2
Abstract

The present invention provides compounds useful as modulators, agonists or antagonists of androgen receptor (AR), compositions thereof, and methods of making and using the same. Compounds of the present invention, and pharmaceutically acceptable compositions thereof, are useful in medicine, and particularly for treating any of a variety of diseases, disorders or conditions.

Claims (9)

1. A compound of formula IV:

or a pharmaceutically acceptable salt thereof, wherein:

X is CH or N;

each R b is independently a substituted or unsubstituted C 1-6 aliphatic; and

n is 0 to 4.

2. The compound according to claim 1 , wherein the compound is:

3. A pharmaceutical composition comprising a compound according to claim 1 , or a pharmaceutically acceptable salt thereof, and a pharmaceutically acceptable carrier, adjuvant, or vehicle.

4. The compound of claim 1 , wherein the compound is represented by the following structural formula:

5. The compound of claim 1 , wherein the compound is represented by the following structural formula:

Assignments (2)
CONFIRMATORY LICENSE Recorded Jun 23, 2016
From: SLOAN-KETTERING INST CAN RESEARCH
To: NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT
Reel/Frame 039121/0139 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Apr 5, 2016
From: BALBAS, MINNA D.; EVANS, MICHAEL J.; SAWYERS, CHARLES L.; SHEN, YANG; HOSFIELD, DAVID; GREENE, GEOFFREY L.
To: MEMORIAL SLOAN-KETTERING CANCER CENTER
Reel/Frame 038190/0833 →
Continuity (2)
Provisional Application 61719117 · Oct 26, 2012
Related Publication 20150274693A1 · Oct 1, 2015