IP Library › Granted Patent US 9,636,413
Granted Patent B2
US 9,636,413 · App. 14/443,212 · Granted May 2, 2017

Conjugates for treating diseases caused by PSMA expressing cells

Inventors: Iontcho Radoslavov Vlahov (West Lafayette, IN); Joseph Anand Reddy (West Lafayette, IN); Alicia Bloomfield (Lafayette, IN); Ryan Dorton (Lafayette, IN); Melissa Nelson (Delphi, IN); Marilynn Vetzel (Rossville, IN); Christopher Paul Leamon (West Lafayette, IN)
Assignee: ENDOCYTE, INC.
A61K47/48246A61K38/05A61K38/06A61K38/07A61K38/08A61K47/48023A61K47/48038A61K49/0002C07K5/021C07K5/06113C07K5/10C07K5/1019A61K38/00
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Quick Facts
Patent No.
US 9,636,413
App. No.
14/443,212
Granted
May 2, 2017
Kind
B2
Abstract

The invention described herein pertains to the diagnosis, imaging, and/or treatment of pathogenic cell populations. In particular, the invention described herein pertains to the diagnosis, imaging, and/or treatment of diseases caused by PSMA expressing cells, such as prostate cancer cells, using compounds capable of targeting PSMA expressing cells.

Claims (12)

1. A conjugate having the formula

or a pharmaceutically acceptable salt thereof.

2. A pharmaceutical composition comprising a conjugate having a formula

or a pharmaceutically acceptable salt thereof.

3. The pharmaceutical composition of claim 2 , wherein the conjugate or the pharmaceutically acceptable salt thereof is present in a therapeutically effective amount for treating a disease in a host animal caused by a pathogenic population of cells, said cells expressing prostate-specific membrane antigen (PSMA).

4. The pharmaceutical composition of claim 2 , further comprising one or a plurality of additional therapeutically active compounds.

5. The pharmaceutical composition of claim 2 , further comprising one or a plurality of pharmaceutically acceptable carriers.

6. The pharmaceutical composition of claim 2 , further comprising one or a plurality of pharmaceutically acceptable diluents.

7. The pharmaceutical composition of claim 2 , further comprising one or a plurality of pharmaceutically acceptable excipients.

8. The pharmaceutical composition of claim 2 , further comprising a component selected from the group consisting of an additional therapeutically active compound, a pharmaceutically acceptable carrier, a pharmaceutically acceptable diluent, a pharmaceutically acceptable excipient, and a combination thereof.

9. The pharmaceutical composition of claim 2 , wherein the pharmaceutical composition is in bulk form.

10. The pharmaceutical composition of claim 2 , e pharmaceutical composition is a unit dose.

Continuity (4)
Provisional Application 61726991 · Nov 15, 2012
Provisional Application 61788382 · Mar 15, 2013
Provisional Application 61875971 · Sep 10, 2013
Related Publication 20150297735A1 · Oct 22, 2015