IP Library Granted Patent US 10,273,202
Granted Patent B2
US 10,273,202 · App. 14/492,741 · Granted Apr 30, 2019

Nitroxyl progenitor compounds and methods of use

Inventors: John P. Toscano (Glen Arm, MD); Christopher M. Pavlos (Laurel, MD); Preeya Kapur Boppana (Frederick, MD)
Assignee: The Johns Hopkins University
C07C247/16C07C247/18C07C291/08C07D207/50C07D209/42
View Patent ↗
Loading inventors, assignments & file history…
Monitor This Case
Get email alerts when status or documents change.
Order Certified Copies
Most orders are placed with the USPTO same day — all within 24 business hours.
Order via The Patent Place →
Pre-filled with this patent's details
Quick Facts
Patent No.
US 10,273,202
App. No.
14/492,741
Granted
Apr 30, 2019
Kind
B2
Abstract

Described herein are nitroxyl progenitor compounds, and compositions including, and methods or generating, the compounds thereof, and methods of treating or preventing disease and disease symptoms using the compounds and compositions.

Claims (9)

1. A compound of formula (I), or a pharmaceutically acceptable salt thereof:

wherein:

R 1 and R 2 , together with the nitrogen to which they are both attached, form a heteroaryl ring, wherein the heteroaryl ring is pyrrolyl or indolyl;

wherein the heteroaryl ring is optionally substituted with from 1-4 groups selected from the group consisting of halo, COOH, NO 2 and ═O;

m is 0; and

n is 0.

2. The compound of claim 1 , or a pharmaceutically acceptable salt thereof, wherein R 1 and R 2 , together with the nitrogen to which they are both attached, form a heteroaryl ring, wherein the heteroaryl ring is substituted with from 1-4 groups selected from the group consisting of halo, COOH, NO 2 and ═O.

3. A compound selected from the group consisting of:

4. A pharmaceutical composition comprising a compound of Formula (I) in claim 1 and a pharmaceutically acceptable carrier.

Assignments (2)
CONFIRMATORY LICENSE Recorded Jan 26, 2018
From: JOHNS HOPKINS UNIVERSITY
To: NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT
Reel/Frame 045169/0607 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jul 28, 2015
From: TOSCANO, JOHN P., III; BOPPANA, PREEYA K.; PAVLOS, CHRISTOPHER M.
To: THE JOHNS HOPKINS UNIVERSITY
Reel/Frame 036196/0620 →
Continuity (4)
Continuation 10587644
Provisional Application 60632456 · Dec 2, 2004
Provisional Application 60540688 · Jan 30, 2004
Related Publication 20150141378A1 · May 21, 2015
Cited By (1)
US 12,186,301