IP Library Granted Patent US 9,107,940
Granted Patent B2
US 9,107,940 · App. 14/508,599 · Granted Aug 18, 2015

Compositions and methods for treating and preventing skeletal muscle deficiencies

Inventors: Rainer Ng (Seattle, WA); Joseph M. Metzger (St. Paul, MN); Lorraine Reeve (Dexter, MI); Bruce Markham (Novi, MI)
Assignees: The Regents of the University of Michigan; Phrixus Pharmaceuticals, Inc.
A61K31/765A61K45/06
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Quick Facts
Patent No.
US 9,107,940
App. No.
14/508,599
Granted
Aug 18, 2015
Kind
B2
Abstract

The present invention relates to compositions and methods for treating and preventing skeletal muscle deficiencies. In particular, the present invention provides compositions comprising poloxamers (e.g., poloxamer 188-P188) and methods of using the same for treating and preventing skeletal muscle deficiencies and injuries (e.g., dystrophin-deficient skeletal muscle; skeletal muscle having a contraction force deficit; skeletal muscle having a Ca 2+ imbalance; skeletal muscle having microtears).

Claims (13)

1. A method of treating or reducing diaphragm skeletal muscle injury or diaphragm skeletal muscle deficiency in a subject comprising administering to a subject in need thereof a composition comprising a therapeutically effective amount of a poloxamer.

2. A methhod of claim 1 , wherein said diaphragm skeletal muscle deficiency is a skeletal muscle contraction force deficit.

3. A method of claim 1 , wherein said poloxamer is a purified or fractionated poloxamer.

4. A method of claim 1 , wherein said subject is a human subject.

5. A method of claim 1 , wherein said composition is administered via intravenous administration.

6. A method of claim 1 , wherein said subject is a dystrophin deficient subject.

7. A method of claim 6 , wherein said subject has Duchene's muscular dystrophy.

8. A method of claim 1 , wherein said treating decreases susceptibility to calcium overload in the diaphragm skeletal muscle of said subject.

9. A method of claim 1 , wherein said poloxamer is P188.

10. A method of claim 1 , wherein said poloxamer is administered at a dosage level of approximately between 0.1-5,000 mg per kg weight of said subject.

11. A method of claim 1 , wherein said poloxamer is administered at a dosage level of approximately between 0.46-500 mg per kg weight of said subject.

12. A method of claim 1 , wherein said dosage level is 0.1-200 mg per kg weight of said subject.

13. A method of claim 1 , wherein said composition comprising a poloxamer is coadministered with one or more agents selected from the group consisting of streptomycin, prednisone, deflazacort, azathioprine, cyclosporine, valproic acid, phenylbutyrate, sodium butyrate, M344, and suberoylanilide hydroxamic acid.

Assignments (3)
CONFIRMATORY LICENSE Recorded Jun 17, 2021
From: UNIVERSITY OF MICHIGAN
To: NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT
Reel/Frame 056575/0663 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Oct 8, 2014
From: REEVE, LORRAINE; MARKHAM, BRUCE
To: PHRIXUS PHARMACEUTICALS, INC.
Reel/Frame 033909/0144 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Oct 8, 2014
From: NG, RAINER; METZGER, JOSEPH M.
To: THE REGENTS OF THE UNIVERSITY OF MICHIGAN
Reel/Frame 033909/0334 →
Continuity (3)
Division 12747073
Provisional Application 61014304 · Dec 17, 2007
Related Publication 20150030559A1 · Jan 29, 2015