IP Library Granted Patent US 9,216,951
Granted Patent B2
US 9,216,951 · App. 14/524,721 · Granted Dec 22, 2015

Lipid-lowering antidiabetic agent

Inventors: Banavara L. Mylari (Lutz, FL); Frank C. Sciavolino (Waterford, CT)
Assignee: Thetis Pharmaceuticals LLC
C07C279/04A61K31/155A61K31/202C07C57/03C07C279/26
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Quick Facts
Patent No.
US 9,216,951
App. No.
14/524,721
Granted
Dec 22, 2015
Kind
B2
Abstract

A composition which includes a salt of metformin and the use of the composition for treatment of or use in prediabetes, diabetes, lowering triglycerides and/or other conditions in mammals.

Claims (10)

1. A method of treating a prediabetic condition in a subject in need thereof, the method comprising administering to the subject a therapeutically effective amount of a pharmaceutical composition comprising a metformin salt of a polyunsaturated fatty acid selected from eicosapentaenoic acid (EPA), docosahexaenoic acid (DHA), and mixtures thereof.

2. The method of claim 1 , wherein the pharmaceutical composition has an aqueous solubility of at least 50 mg/ml under standard conditions.

3. The method of claim 1 , wherein the subject has serum triglyceride levels of greater than 200 mg/dl.

4. The method of claim 1 , wherein the subject has hypertriglyceridemia.

5. The method of claim 1 , wherein the metformin salt of a polyunsaturated fatty acid is a polymorph, solvate, or hydrate.

6. The method of claim 1 , wherein the subject is further selected from the group consisting of subjects having or at risk of developing diabetes, a prediabetic condition, obesity, cardiac arrhythmia, myocardial infarction, and stroke due to high serum triglyceride levels.

7. The method of claim 1 , wherein the prediabetic condition is incipient diabetes with impaired glucose tolerance.

8. The method of claim 1 , wherein the polyunsaturated fatty acid is eicosapentaenoic acid (EPA).

9. The method of claim 1 , wherein the polyunsaturated fatty acid is docosahexaenoic acid (DHA).

10. The method of claim 1 , wherein the polyunsaturated fatty acid is a mixture of EPA and DHA.

Assignments (2)
SECURITY AGREEMENT Recorded Aug 17, 2018
From: THETIS PHARMACEUTICALS LLC
To: CONNECTICUT INNOVATIONS, INC., AS COLLATERAL AGENT
Reel/Frame 046850/0287 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Oct 28, 2014
From: MYLARI, BANAVARA L., MR.; SCIAVOLINO, FRANK C., MR.
To: THETIS PHARMACEUTICALS LLC
Reel/Frame 034047/0169 →
Continuity (4)
Continuation 13923829 · Jun 21, 2013
Division 13348265 · Jan 11, 2012
Provisional Application 61461113 · Jan 12, 2011
Related Publication 20150051284A1 · Feb 19, 2015