IP Library Granted Patent US 9,682,123
Granted Patent B2
US 9,682,123 · App. 14/579,913 · Granted Jun 20, 2017

Methods of treating metabolic disease

Inventors: Rudolph L. Leibel (New York, NY); Kazuhisa Watanabe (Shimotsuke, JP); Wendy K. Chung (Hackensack, NJ); Stuart G. Fischer (New Rochelle, NY); Charles Leduc (Hackensack, NJ); Elizabeth Watson (New York, NY); Maria Laura Cremona (Englewood, NJ)
Assignee: THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK
A61K38/1774A01K67/0276A61K31/00A61K31/713A61K31/7105A61K45/06C07K14/70503A01K2217/075A01K2217/206A01K2227/105A01K2267/0362A61K48/00
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Quick Facts
Patent No.
US 9,682,123
App. No.
14/579,913
Granted
Jun 20, 2017
Kind
B2
Abstract

The invention provides methods for treating metabolic disease in a subject and methods for increasing the expression of ILDR2 in a subject. The invention further provides a method for identifying an agent which modulates expression of an Ildr2 RNA comprising contacting a cell with an agent; determining expression of the Ildr2 RNA in the presence and the absence of the agent; and comparing expression of the Ildr2 RNA in the presence and the absence of the agent, wherein a change in the expression of the Ildr2 RNA in the presence of the agent is indicative of an agent which modulates the level of expression of the RNA.

Claims (15)

1. A method of treating hepatic steatosis in a subject, the method comprising administering to the subject a therapeutically effective amount of an adenoviral expression vector comprising a nucleic acid encoding full-length ILDR2, and wherein the subject has metabolic syndrome, type II diabetes, insulin resistance, or is obese, or any combination thereof.

2. A method of decreasing hepatic triglyceride level or hepatic total cholesterol level in a subject, the method comprising administering to the subject a therapeutically effective amount of an adenoviral expression vector comprising a nucleic acid encoding full-length ILDR2.

3. The method of claim 2 , wherein the hepatic triglyceride level or hepatic total cholesterol level is decreased relative to a hepatic triglyceride level or hepatic total cholesterol level in the subject before administrating the therapeutically effective amount of an adenoviral expression vector comprising a nucleic acid encoding full-length ILDR2.

4. The method of claim 1 or 2 , wherein the expression of Ildr2 mRNA or ILDR2 protein is increased in liver tissue.

5. The method of claim 1 or 2 , wherein the expression of Ildr2 mRNA or ILDR2 protein is increased in hepatocytes.

6. The method of claim 1 or 2 , wherein the subject is administered an additional therapy.

7. The method of claim 6 , wherein the additional therapy is a lipid lowering therapy.

8. The method of claim 7 , wherein the lipid lowering therapy is a therapeutic lifestyle change, a HMG-CoA reductase inhibitor, niacin, a fibrate, a cholesterol absorption inhibitor, a MTP inhibitor, or any combination thereof.

9. The method of claim 1 or 2 , wherein expression of ILDR2 protein in the subject is measured using an antibody.

10. The method of claim 9 , wherein the antibody specifically binds to a peptide selected from the group consisting of SEQ ID NOs: 2-9, an ILDR2 protein, or an ILDR2 isoform.

11. The method of claim 1 , wherein the subject has a reduced level of expression of Ildr2 mRNA or ILDR2 protein compared to the level of expression of Ildr2 mRNA or ILDR2 protein in a subject without hepatic steatosis.

12. The method of claim 9 , wherein the level of expression is determined before administrating to the subject the therapeutically effective amount of an adenoviral expression vector comprising a nucleic acid encoding full-length ILDR2.

13. The method of claim 11 , wherein the expression of ILDR2 protein in the subject is measured using an antibody.

14. The method of claim 13 , wherein the antibody specifically binds to a peptide selected from the group consisting of SEQ ID NOs: 2-9, an ILDR2 protein, or an ILDR2 isoform.

15. A method of decreasing liver fat deposits in a subject, the method comprising administering to the subject a therapeutically effective amount of an adenoviral expression vector comprising a nucleic acid encoding full-length ILDR2.

Assignments (3)
CONFIRMATORY LICENSE Recorded Aug 23, 2023
From: THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK
To: NATIONAL INSTITUTES OF HEALTH - DIRECTOR DEITR
Reel/Frame 064686/0180 →
CONFIRMATORY LICENSE Recorded Aug 23, 2017
From: COLUMBIA UNIV NEW YORK MORNINGSIDE
To: NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT
Reel/Frame 043644/0845 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Feb 24, 2015
From: LEIBEL, RUDOLPH L; WATANABE, KAZUHISA; CHUNG, WENDY K; FISCHER, STUART G; LEDUC, CHARLES; WATSON, ELIZABETH; CREMONA, MARIA LAURA
To: THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK
Reel/Frame 035019/0249 →
Continuity (2)
Provisional Application 61919367 · Dec 20, 2013
Related Publication 20150190466A1 · Jul 9, 2015