IP Library › Granted Patent US 9,526,728
Granted Patent B2
US 9,526,728 · App. 14/633,489 · Granted Dec 27, 2016

Medical use of a DPP-4 inhibitor

Inventors: Thomas Klein (Radolfzell, DE); Andrew Advani (Toronto, CA); Kim Alexander Connelly (Toronto, CA); Richard Ernest Gilbert (Toronto, CA)
Assignee: Boehringer Ingelheim International GmbH
A61K31/519A61K31/155A61K31/4439A61K31/4985A61K31/522A61K31/64A61K45/06
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Quick Facts
Patent No.
US 9,526,728
App. No.
14/633,489
Granted
Dec 27, 2016
Kind
B2
Abstract

The present invention relates to the use of 1-[(4-methyl-quinazolin-2-yl)methyl]-3 -methyl-7-(2-butyn-1-yl)-8-(3-(R)-amino-piperidin-1-yl)-xanthine for use in a patient being at risk of or having heart failure with preserved ejection fraction (HFpEF).

Claims (8)

1. A method for treating a patient being at risk of or having heart failure with preserved ejection fraction (HFpEF), the method comprising administering to the patient 1-[(4-methyl-quinazolin-2-yl)methyl]-3-methyl-7-(2-butyn-1-yl)-8-(3-(R)-amino-piperidin-1-yl)-xanthine, optionally in combination with one or more other active agents.

2. The method of claim 1 , wherein the patient has chronic kidney disease (CKD).

3. The method of claim 1 , wherein the patient has severe renal impairment or end-stage renal disease (ESRD).

4. The method of claim 1 , said method further comprising treating, reducing the risk of, slowing progression of, delaying the onset of, and/or protecting against heart failure with preserved ejection fraction (HFpEF) and/or diseases associated therewith.

5. The method of claim 4 , wherein the disease associated with HFpEF is a major adverse cardiovascular event (MACE) selected from the group consisting of myocardial infarction, stroke, cardiovascular death, and cardiovascular hospitalization for unstable or stable angina pectoris, heart failure and coronary revascularization.

6. The method of claim 1 , said method further comprising treating, reducing the risk of, slowing progression of, delaying the onset of, and/or protecting against diastolic dysfunction and/or cardiac fibrosis.

7. The method of claim 1 , wherein the patient is a diabetic patient.

8. The method of claim 1 , wherein the patient is a non-diabetic patient.

Assignments (1)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Apr 7, 2015
From: KLEIN, THOMAS; ADVANI, ANDREW; CONNELLY, KIM ALEXANDER; GILBERT, RICHARD ERNEST
To: BOEHRINGER INGELHEIM INTERNATIONAL GMBH
Reel/Frame 035345/0320 →
Priority Claims (1)
EP 14157222 · Feb 28, 2014 · regional
Continuity (1)
Related Publication 20150246045A1 · Sep 3, 2015