IP Library › Granted Patent US 9,345,680
Granted Patent B2
US 9,345,680 · App. 14/671,585 · Granted May 24, 2016

Compounds and their salts specific to the PPAR receptors and the EGF receptors and their use in the medical field

Inventors: Giancarlo Naccari (Monza, IT); Sergio Baroni (Villa D'adda, IT)
Assignee: Nogra Pharma Limited
A61K31/196C07C229/42
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Quick Facts
Patent No.
US 9,345,680
App. No.
14/671,585
Granted
May 24, 2016
Kind
B2
Abstract

The present invention relates to compounds comprising the general formula (I), in which R 1 and R 2 , which may be identical or different, are selected from the group comprising —H or a linear or branched alkyl group having from 1 to 6 carbon atoms or together form an aromatic or aliphatic ring with 5 or 6 atoms; Y and Z, which may be identical or different, are selected from the group comprising —H, —OH, —COOH, —OR 3 , —CH(OR 3 )COOH, in which R 3 is selected from H, phenyl, benzyl, —CF 3 or —CF 2 CF 3 , vinyl, allyl and a linear or branched alkyl group having from 1 to 6 carbon atoms.

Claims (10)

1. A pharmaceutical composition comprising (R)-2-methoxy-3-(4′-aminophenyl)propionic acid, or a pharmaceutically acceptable salt thereof; and a pharmaceutically acceptable excipient.

2. A method of treating a chronic inflammatory disease selected from the group consisting of Crohn's disease and ulcerative rectocolitis, comprising administering to a mammal in need thereof the pharmaceutical composition of claim 1 .

3. The method of claim 2 , wherein the disease is Crohn's disease.

4. The method of claim 2 , wherein the disease is ulcerative rectocolitis.

5. The method of claim 2 , wherein the mammal is a human.

6. A pharmaceutical composition comprising (S)-2-methoxy-3-(4′-aminophenyl)propionic acid, or a pharmaceutically acceptable salt thereof; and a pharmaceutically acceptable excipient.

7. A method of treating a chronic inflammatory disease selected from the group consisting of Crohn's disease and ulcerative rectocolitis, comprising administering to a mammal in need thereof the pharmaceutical composition of claim 6 .

8. The method of claim 7 , wherein the disease is Crohn's disease.

9. The method of claim 7 , wherein the disease is ulcerative rectocolitis.

10. The method of claim 7 , wherein the mammal is a human.

Assignments (2)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Apr 27, 2016
From: NACCARI, GIANCARLO; BARONI, SERGIO
To: GIULIANI INTERNATIONAL LIMITED
Reel/Frame 038394/0536 →
CHANGE OF NAME Recorded Apr 27, 2016
From: GIULIANI INTERNATIONAL LIMITED
To: NOGRA PHARMA LIMITED
Reel/Frame 038538/0485 →
Priority Claims (1)
IT RM2005A0389 · Jul 22, 2005 · national
Continuity (4)
Continuation 14202386 · Mar 10, 2014
Continuation 13408439 · Feb 29, 2012
Division 11989090
Related Publication 20150265563A1 · Sep 24, 2015