IP Library Granted Patent US 10,098,903
Granted Patent B2
US 10,098,903 · App. 14/700,232 · Granted Oct 16, 2018

Inhibiting inflammation with milk oligosaccharides

Inventors: Ardythe L. Morrow (Cincinnati, OH); David S. Newburg (Newtonville, MA); Guillermo M. Ruiz-Palacios (Mexico City, MX)
Assignees: Children's Hospital Medical Center; The General Hospital Corporation; Instituto Nacional de Ciencias Medicas Y Nutricion
A61K31/7016A61K31/702A61K47/62A61K35/20A61K47/50A61K47/61
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Quick Facts
Patent No.
US 10,098,903
App. No.
14/700,232
Granted
Oct 16, 2018
Kind
B2
Abstract

A method of inhibiting inflammation with milk oligosaccharides or glycoconjugates containing the oligosaccharides.

Claims (35)

1. A method of treating ulcerative colitis, Crohn's disease, or irritable bowel syndrome, comprising administering to a subject in need thereof an effective amount of a composition consisting essentially of one or more human milk-derived oligosaccharides, wherein at least one of the one or more human milk-derived oligosaccharides is selected from the group consisting of:

(i) 3-Fucosyllactose (3-FL),

(ii) Lacto-N-fucopentaose I (LNF-I),

(iii) Lactodifucotetraose (LDFT),

(iv) Lacto-N-neotetraose, and

(v) Lacto-N-tetraose.

2. The method of claim 1 , wherein the human milk-derived oligosaccharide is conjugated with a carbohydrate, a lipid, a polypeptide, or a peptide to form a glycoconjugate.

3. The method of claim 1 , wherein the subject suffers from or is at risk for ulcerative colitis, Crohn's disease, or irritable bowel syndrome.

4. The method of claim 1 , wherein the composition is formulated for oral administration.

5. The method of claim 4 , wherein the composition further contains a pharmaceutically acceptable carrier and a lubricating agent.

6. The method of claim 4 , wherein the composition further contains a sweetening agent, a flavoring agent, a coloring agent, or a combination thereof.

7. The method of claim 1 , wherein the one or more human milk-derived oligosaccharides are synthesized chemically, isolated from milk, or produced by a microorganism.

8. The method of claim 1 , wherein the composition is formulated as a food product or food supplement.

9. The method of claim 1 , wherein the one or more human milk-derived oligosaccharides further comprise 2′-fucosyllactose.

10. The method of claim 9 , wherein the one or more human milk-derived oligosaccharides consists of 2′-fucosyllactose and lacto-N-neotetraose.

11. The method of claim 10 , wherein the composition is formulated for oral administration.

12. The method of claim 10 , wherein the subject is a human patient having irritable bowel syndrome.

13. The method of claim 10 , wherein the composition further contains a pharmaceutically acceptable carrier.

14. The method of claim 13 , wherein the pharmaceutically acceptable carrier is silicon dioxide.

15. The method of claim 1 , wherein the one or more human milk-derived oligosaccharides are free oligosaccharides.

16. A method of treating ulcerative colitis, Crohn's disease, or irritable bowel syndrome, comprising administering to a subject in need thereof an effective amount of a composition comprising an agent that inhibits inflammation and a pharmaceutically acceptable carrier, wherein the agent is the only agent that inhibits inflammation, and consists of one or more human milk-derived oligosaccharides, and wherein at least one of the one or more human milk-derived oligosaccharides is selected from the group consisting of:

(i) 3-Fucosyllactose (3-FL),

(ii) Lacto-N-fucopentaose I (LNF-I),

(iii) Lactodifucotetraose (LDFT),

(iv) Lacto-N-neotetraose, and

(v) Lacto-N-tetraose.

17. The method of claim 16 , wherein the one or more human milk-derived oligosaccharides further comprise 2′-fucosyllactose.

18. The method of claim 17 , wherein the one or more human milk-derived oligosaccharides comprise 2′-fucosyllactose and lacto-N-neotetraose.

19. The method of claim 17 , wherein the agent that inhibits inflammation consists of 2′-fucosyllactose and lacto-N-neotetraose.

20. The method of claim 16 , wherein the composition consists of the agent that inhibits inflammation and the pharmaceutically acceptable carrier.

21. The method of claim 16 , wherein the composition is formulated for oral administration.

22. The method of claim 16 , wherein the pharmaceutically acceptable carrier comprises silicon dioxide.

23. The method of claim 16 , wherein the subject is a human patient having irritable bowel syndrome.

24. The method of claim 16 , wherein the one or more human milk-derived oligosaccharides are synthesized chemically, isolated from milk, or produced by a microorganisms.

25. The method of claim 16 , wherein the one or more human milk-derived oligosaccharides are free oligosaccharides.

Assignments (4)
CONFIRMATORY LICENSE Recorded Sep 23, 2019
From: CINCINNATI CHILDREN'S HOSPITAL MEDICAL CENTER
To: NATIONAL INSTITUTES OF HEALTH -DIRECTOR DEITR
Reel/Frame 050460/0048 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Nov 10, 2015
From: NEWBURG, DAVID S.
To: THE GENERAL HOSPITAL CORPORATION D/B/A MASSACHUSETTS GENERAL HOSPITAL
Reel/Frame 036999/0536 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Nov 10, 2015
From: RUIZ-PALACIOS, GUILLERMO
To: INSTITUTO NACIONAL DE CIENCIAS MEDICAS Y NUTRICION
Reel/Frame 036999/0627 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jun 1, 2015
From: MORROW, ARDYTHE
To: CHILDREN'S HOSPITAL MEDICAL CENTER
Reel/Frame 035753/0556 →
Continuity (3)
Continuation 13382323
Provisional Application 61223145 · Jul 6, 2009
Related Publication 20150306120A1 · Oct 29, 2015
Cited By (2)
US 12,364,721 US 12,383,569