IP Library Granted Patent US 9,492,554
Granted Patent B2
US 9,492,554 · App. 14/703,549 · Granted Nov 15, 2016

Methods and compositions related to viral inhibition

Inventors: Dev P. Arya (Greenville, SC); Nihar Ranjan (Clemson, SC); Sunil Kumar (Clemson, SC)
Assignee: Clemson University
A61K47/48061
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Quick Facts
Patent No.
US 9,492,554
App. No.
14/703,549
Granted
Nov 15, 2016
Kind
B2
Abstract

Disclosed herein are compounds, compositions and methods related to viral inhibition. In some forms, the compounds, compositions and methods are related to binding RNA.

Claims (36)

1. A method of inhibiting a viral life cycle, comprising incubating a virus with a composition wherein said composition comprises a compound comprising the structure

A-B-C

or a pharmaceutically acceptable salt or acid form thereof,

wherein A is a glycoside, aminoglycoside, or sugar,

wherein B is a linker defined by -(L 1 ) v -, wherein v is independently 1-20,

wherein each (L 1 ) is independently O, N, S, C 1 -C 8 alkyl, C 2 -C 8 alkenyl, C 2 -C 8 alkoxy, aryl, heteroaryl, heterocyclyl,

wherein each (L1) is the same or different, and

wherein C is a glycoside, aminoglycoside, sugar, Hoechst 33258, or a benzimidazole.

2. A method of treating a disease, comprising administering to a subject a composition comprising a compound comprising the structure

A-B-C

or a pharmaceutically acceptable salt or acid form thereof,

wherein A is a glycoside, aminoglycoside, or sugar,

wherein B is a linker defined by -(L 1 ) v -, wherein v is independently 1-20,

wherein each (L 1 ) is independently O, N, S, C 1 -C 8 alkyl, C 2 -C 8 alkenyl, C 2 -C 8 alkoxy, aryl, heteroaryl, heterocyclyl,

wherein each (L1) is the same or different, and wherein C is a glycoside, aminoglycoside, sugar, Hoechst 33258, or a benzimidazole.

3. The method of claim 2 , wherein the disease is a viral disease.

4. A method of protecting cells from HIV cytopathic effects, comprising contacting a cell with a composition comprising a compound comprising the structure

A-B-C

or a pharmaceutically acceptable salt or acid form thereof,

wherein A is a glycoside, aminoglycoside, or sugar,

wherein B is a linker defined by -(L 1 ) v -, wherein v is independently 1-20,

wherein each (L 1 ) is independently O, N, S, C 1 -C 8 alkyl, C 2 -C 8 alkenyl, C 2 -C 8 alkoxy, aryl, heteroaryl, heterocyclyl,

wherein each (L1) is the same or different, and wherein C is a glycoside, aminoglycoside, sugar, Hoechst 33258, or a benzimidazole.

5. The method of claim 4 , wherein the cell is in vivo in a subject.

6. The method of inhibiting a viral life cycle of claim 1 wherein said A is an aminoglycoside.

7. The method of inhibiting a viral life cycle of claim 6 wherein said A comprises neomycin.

8. The method of inhibiting a viral life cycle of claim 1 wherein said B comprises a backbone of less than 50.

9. The method of inhibiting a viral life cycle of claim 1 wherein said benzimidazole is a Hoechst 33258 derived benzimidazole.

10. The method of treating a disease of claim 2 wherein said A is an aminoglycoside.

11. The method of treating a disease of claim 10 wherein said A comprises neomycin.

12. The method of treating a disease of claim 2 wherein said B comprises a backbone of less than 50.

13. The method of treating a disease of claim 2 wherein said benzimidazole is a Hoechst 33258 derived benzimidazole.

14. The method of protecting cells from HIV cytopathic effects of claim 4 wherein said A is an aminoglycoside.

15. The method of protecting cells from HIV cytopathic effects claim 14 wherein said A comprises neomycin.

16. The method of protecting cells from HIV cytopathic effects claim 4 wherein said B comprises a backbone of less than 50.

17. The method of protecting cells from HIV cytopathic effects claim 4 wherein said benzimidazole is a Hoechst 33258 derived benzimidazole.

Assignments (3)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jun 28, 2016
From: ARYA, DEV P.; RANJAN, NIHAR; KUMAR, SUNIL
To: CLEMSON UNIVERSITY
Reel/Frame 039026/0908 →
CONFIRMATORY LICENSE Recorded Sep 3, 2015
From: CLEMSON UNIVERSITY
To: NATIONAL SCIENCE FOUNDATION
Reel/Frame 036539/0121 →
CONFIRMATORY LICENSE Recorded May 29, 2015
From: CLEMSON UNIVERSITY
To: NATIONAL SCIENCE FOUNDATION
Reel/Frame 035802/0236 →
Continuity (4)
Division 12857425 · Aug 16, 2010
Provisional Application 61234260 · Aug 14, 2009
Provisional Application 61234603 · Aug 17, 2009
Related Publication 20160263231A1 · Sep 15, 2016