IP Library Granted Patent US 10,927,192
Granted Patent B2
US 10,927,192 · App. 14/709,674 · Granted Feb 23, 2021

Composition and method of making water soluble chitosan polymer and composite particles

Inventors: Santra Swadeshmukul (Orlando, FL); Basumallick Srijita (Orlando, FL)
Assignee: University of Central Florida Research Foundation, Inc.
C08B37/003A01N55/02A01N59/20A61K9/5161A61K9/5192A61K47/36A61L15/24A61L15/28A61L15/46A61L26/0014A61L26/0023A61L26/0066A61L27/16A61L27/20A61L27/54A61L31/042A61L31/048A61L31/16
View Patent ↗
Loading inventors, assignments & file history…
Monitor This Case
Get email alerts when status or documents change.
Order Certified Copies
Most orders are placed with the USPTO same day — all within 24 business hours.
Order via The Patent Place →
Pre-filled with this patent's details
Quick Facts
Patent No.
US 10,927,192
App. No.
14/709,674
Granted
Feb 23, 2021
Kind
B2
Abstract

Embodiments of the present disclosure provide for water-soluble chitosan particles, methods of making water-soluble chitosan particles, and methods of using water-soluble chitosan particles. In an embodiment, the composition of water-soluble chitosan particles can be used in drug delivery, tissue engineering, bioimaging, biosensing, catalysis, and antimicrobial applications.

Claims (20)

1. A composition comprising: a water-soluble chitosan nanoparticle, wherein the water-soluble chitosan nanoparticle comprises an ionic complex of a composite of a bicarboxylic acid compound, a metal oxide having mixed valence states and a depolymerized chitosan, the depolymerized chitosan comprising chitosan oligomers, chitosan monomers, or a combination thereof wherein each chitosan component of the depolymerized chitosan has a molecular weight that is less than 50,000 Da.

2. The composition of claim 1 , wherein the bicarboxylic acid compound is selected from the group consisting tartaric acid, malic acid, succinic acid, and a combination thereof.

3. The composition of claim 1 , wherein the metal oxide is bonded within the composite of the depolymerized chitosan and the bicarboxylic acid compound.

4. The composition of claim 1 , wherein the metal oxide is is oxide of copper.

5. The composition of claim 4 , wherein copper in the metal oxide has an oxidation state of a combination of Cu(I), Cu(II).

6. The composition of claim 4 , wherein the water-soluble chitosan nanoparticle has antimicrobial properties.

7. The composition of claim 4 , wherein the metal oxide is not separately water soluble, while the water soluble chitosan nanoparticle and the metal oxide combination is water soluble.

8. A method of making a composition, comprising:

mixing a chitosan polymer, a metal oxide having mixed valence states and a bicarboxylic acid compound, the chitosan polymer having a molecular weight of from about 50,000 Da to about 190,000 Da; and hydrothermal treating of the mixture to form a water-soluble chitosan nanoparticle, wherein the temperature utilized in the hydrothermal treatment is about 135 to 150° C., and the pressure of the hydrothermal treatment is greater than 1 atm and up to 5 atm, the water-soluble chitosan nanoparticle comprises a composite of a bicarboxylic acid compound and a depolymerized chitosan, the depolymerized chitosan comprising chitosan oligomers, chitosan monomers, or a combination thereof, wherein each chitosan component of the depolymerized chitosan has a molecular weight that is less than 50,000 Da.

9. The method of claim 8 , wherein the bicarboxylic acid compound is selected from the group consisting of: tartaric acid, malic acid, succinic acid, and a combination thereof.

10. The method of claim 8 , wherein the metal oxides are oxides of copper.

11. The method of claim 10 , wherein copper is selected from a combination of Cu(I), Cu(II).

12. The composition of claim 1 , wherein a weight ratio of the depolymerized chitosan and the bicarboxylic acid compound in the composite of the water-soluble chitosan nanoparticle is from 2:1 to 2.5:1.

13. The composition of claim 1 , wherein the water-soluble chitosan nanoparticle is a hydrothermally-treated water-soluble chitosan nanoparticle, wherein the water-soluble chitosan nanoparticle has a diameter of about 10 nm to about 100 nm.

14. The composition of claim 13 , wherein the water-soluble chitosan nanoparticle has a diameter of about 30 nm to about 50 nm.

15. The composition of claim 1 , wherein the depolymerized chitosan of the water-soluble chitosan nanoparticle is defined by a cleavage at a glycoside linkage of a chitosan precursor, the cleavage at the glycoside linkage being confirmed by a Fourier Transform Infrared Spectrum.

16. The composition of claim 3 , wherein the metal oxide comprises a metal oxide nanoparticle.

17. The method of claim 8 , wherein the mixing comprises mixing the chitosan polymer and the bicarboxylic acid compound in a weight proportion of about 0.8:1.2 to about 1.2:0.8.

18. The method of claim 17 , wherein the mixing further comprises mixing the chitosan polymer and the bicarboxylic acid compound in a weight proportion of about 1:1.

19. The method of claim 8 , wherein the pressure of the hydrothermal treatment is about 2.5 atm.

Assignments (3)
CONFIRMATORY LICENSE Recorded Nov 16, 2017
From: UNIVERSITY OF CENTRAL FLORIDA
To: NATIONAL SCIENCE FOUNDATION
Reel/Frame 044479/0894 →
CORRECTIVE ASSIGNMENT TO CORRECT THE NAME OF THE ASSIGNEE PREVIOUSLY RECORDED AT REEL: 036290 FRAME: 0897. ASSIGNOR(S) HEREBY CONFIRMS THE ASSIGNMENT. Recorded Sep 28, 2016
From: SANTRA, SWADESHMUKUL; BASUMALLICK, SRIJITA
To: UNIVERSITY OF CENTRAL FLORIDA RESEARCH FOUNDATION, INC.
Reel/Frame 040171/0099 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Aug 10, 2015
From: SANTRA, SWADESHMUKUL; BASUMALLICK, SRIJITA
To: UNIVERSITY OF CENTRAL FLORIDA RESEARCH FOUNDATION INC.
Reel/Frame 036290/0897 →
Continuity (2)
Provisional Application 61992510 · May 13, 2014
Related Publication 20150327553A1 · Nov 19, 2015