IP Library Granted Patent US 9,604,962
Granted Patent B2
US 9,604,962 · App. 14/748,372 · Granted Mar 28, 2017

Fungicidal azocyclic amides

Inventors: Robert James Pasteris (Newark, DE); Rafael Shapiro (Wilmington, DE)
Assignee: E I DU PONT DE NEMOURS AND COMPANY
C07D401/06A01N43/78A01N43/80C07D211/62C07D231/12C07D261/04C07D261/08C07D413/14C07D417/14
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Quick Facts
Patent No.
US 9,604,962
App. No.
14/748,372
Granted
Mar 28, 2017
Kind
B2
Abstract

Disclosed are compounds of Formulae 1, 1A, 1B and 1C including all geometric and stereoisomers, N-oxides, and salts thereof, wherein R 1 , R 2 , R 4a1 , R 4a2 , A, A a , G, M, W, Z 1 , Z 3 , X, J, J 1 and n are as defined in the disclosure. Also disclosed are compositions containing the compounds of Formula 1 and methods for controlling plant disease caused by a fungal pathogen comprising applying an effective amount of a compound or a composition of the invention.

Claims (14)

1. A compound selected from Formula 1B, an N-oxide and salt thereof

wherein

each R 4a1 and R 4a2 is independently C 1 -C 3 alkyl, C 2 -C 3 alkenyl, C 2 -C 3 alkynyl, cyclopropyl, C 1 -C 3 haloalkyl, C 2 -C 3 haloalkenyl, C 2 -C 3 haloalkynyl, halocyclopropyl, halogen, cyano, nitro, C 1 -C 2 alkoxy, C 1 -C 2 haloalkoxy, C 1 -C 2 alkylthio, C 1 -C 2 haloalkylthio, C 2 -C 3 alkoxyalkyl, C 2 -C 3 alkylcarbonyl, C 2 -C 3 alkoxycarbonyl, C 2 -C 3 alkylaminocarbonyl or C 3 -C 4 dialkylaminocarbonyl; and

Z 3 is CN or C(═S)NH 2 .

2. A compound of claim 1 wherein

each R 4a1 and R 4a2 is independently C 1 -C 3 alkyl, C 1 -C 3 haloalkyl, halogen, cyano, C 1 -C 2 alkoxy or C 1 -C 2 haloalkoxy.

3. A compound of claim 1 selected from the group consisting of:

1-[2-[5-methyl-3-(trifluoromethyl)-1H-pyrazol-1-yl]acetyl]-4-piperidinecarbothioamide,

1-[2-[3,5-bis(trifluoromethyl)-1H-pyrazol-1-yl]acetyl]-4-piperidinecarbothioamide,

1-[2-[5-methyl-3-(trifluoromethyl)-1H-pyrazol-1-yl]acetyl]-4-piperidinecarbonitrile, and

1-[2-[3,5-bis(trifluoromethyl)-1H-pyrazol-1-yl]acetyl]-4-piperidinecarbonitrile.

4. A compound selected from:

1-(2-chloroacetyl)-4-piperidinecarbonitrile and

1-(2-chloroacetyl)-N-(1,1-dimethylethyl)-4-piperidinecarboxamide.

Assignments (1)
NUNC PRO TUNC ASSIGNMENT Recorded Nov 29, 2022
From: E.I. DU PONT DE NEMOURS AND COMPANY
To: CORTEVA AGRISCIENCE LLC
Reel/Frame 063141/0155 →
Continuity (6)
Division 14087481 · Nov 22, 2013
Division 12303256
Continuation In Part PCTUS2007014647 · Jun 22, 2007
Provisional Application 60833824 · Jul 27, 2006
Provisional Application 60897173 · Jan 24, 2007
Related Publication 20150291556A1 · Oct 15, 2015