IP Library › Granted Patent US 9,694,016
Granted Patent B2
US 9,694,016 · App. 14/774,431 · Granted Jul 4, 2017

Biaryl amide compounds as kinase inhibitors

Inventors: Robert John Aversa (Watertown, MA); Paul Andrew Barsanti (Pleasant Hill, CA); Matthew Burger (Belmont, MA); Michael Patrick Dillon (Boston, MA); Alan Dipesa (Bronx, NY); Cheng Hu (San Mateo, CA); Yan Lou (Pleasanton, CA); Gisele Nishiguchi (Arlington, MA); Yue Pan (Lexington, MA); Valery Polyakov (Moraga, CA); Savithri Ramurthy (Arlington, MA); Alice Rico (Castro Valley, CA); Lina Setti (Fremont, CA); Aaron Smith (Fremont, CA); Sharadha Subramanian (San Ramon, CA); Benjamin Taft (Oakland, CA); Huw Tanner (San Francisco, CA); Lifeng Wan (Union City, CA); Naeem Yusuff (Cambridge, MA)
Assignee: NOVARTIS AG
A61K31/5377A61K31/5375A61K31/541A61K45/06C07D213/74C07D213/75C07D213/81C07D213/82C07D213/84C07D233/88C07D237/20C07D237/22C07D239/42C07D239/47C07D239/48C07D241/20C07D263/58C07D277/42C07D401/04C07D401/12C07D401/14C07D403/04C07D403/12C07D405/04C07D405/12C07D405/14C07D409/14C07D413/04C07D413/12C07D413/14C07D417/12C07D471/04C07D487/04C07D491/048C07D491/107C07D493/04C07D493/10C07D495/04C07D498/08C07D513/04
View Patent ↗
Loading inventors, assignments & file history…
Monitor This Case
Get email alerts when status or documents change.
Order Certified Copies
Most orders are placed with the USPTO same day — all within 24 business hours.
Order via The Patent Place →
Pre-filled with this patent's details
Quick Facts
Patent No.
US 9,694,016
App. No.
14/774,431
Granted
Jul 4, 2017
Kind
B2
Abstract

The present invention provides compounds of Formula (I) as described herein, and salts thereof, and therapeutic uses of these compounds for treatment of disorders associated with Raf kinase activity. The invention further provides pharmaceutical compositions comprising these compounds, and compositions comprising these compounds and a therapeutic co-agent.

Claims (13)

1. A compound, or a pharmaceutically acceptable salt thereof, selected from:

2. A pharmaceutical composition comprising a compound of claim 1 or a pharmaceutically acceptable salt thereof and one or more pharmaceutically acceptable carriers.

3. A combination comprising a therapeutically effective amount of a compound according to claim 1 or a pharmaceutically acceptable salt thereof and one or more therapeutically active co-agents.

4. The compound according to claim 1 that is:

or a pharmaceutically acceptable salt thereof.

5. The compound according to claim 1 that is:

or a pharmaceutically acceptable salt thereof.

6. The compound according to claim 1 that is:

or a pharmaceutically acceptable salt thereof.

7. The compound according to claim 1 that is:

or a pharmaceutically acceptable salt thereof.

8. The compound according to claim 1 that is:

or a pharmaceutically acceptable salt thereof.

Assignments (5)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Oct 23, 2015
From: AVERSA, ROBERT; BARSANTI, PAUL A.; BURGER, MATTHEW; DILLON, MICHAEL PATRICK; HU, CHENG; LOU, YAN; NISHIGUCHI, GISELE; PAN, YUE; POLYAKOV, VALERY; RAMURTHY, SAVITHRI; RICO, ALICE; SETTI, LINA; SMITH, AARON; SUBRAMANIAN, SHARADHA; TAFT, BENJAMIN; TANNER, HUW; WAN, LIFENG
To: NOVARTIS VACCINES AND DIAGNOSTICS, INC.
Reel/Frame 036865/0210 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Oct 23, 2015
From: DIPESA, ALAN
To: NOVARTIS INSTITUTES FOR BIOMEDICAL RESEARCH INC.
Reel/Frame 036865/0369 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Oct 23, 2015
From: YUSUFF, NAEEM
To: NOVARTIS INSTITUTES FOR BIOMEDICAL RESEARCH INC.
Reel/Frame 036865/0390 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Oct 23, 2015
From: NOVARTIS VACCINES AND DIAGNOSTICS, INC.
To: NOVARTIS AG
Reel/Frame 036865/0419 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Oct 23, 2015
From: NOVARTIS INSTITUTES FOR BIOMEDICAL RESEARCH INC.
To: NOVARTIS AG
Reel/Frame 036865/0436 →
Continuity (2)
Provisional Application 61783558 · Mar 14, 2013
Related Publication 20160038504A1 · Feb 11, 2016