IP Library Granted Patent US 9,446,152
Granted Patent B2
US 9,446,152 · App. 14/838,586 · Granted Sep 20, 2016

Polyethylene glycol based oligomers for coating nanoparticles, nanoparticles coated therewith, and related methods

Inventors: Hedi Mattoussi (Tallahassee, FL); Goutam Palui (Tallahassee, FL); Hyon Bin Na (Seoul, KR)
Assignee: The Florida State University Research Foundation, Inc.
A61K49/0067C08F8/32C08F20/06C08F22/00C08K5/00C08K5/13C08L33/00C08L71/08C09D133/14H01F1/0054C08F220/26
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Quick Facts
Patent No.
US 9,446,152
App. No.
14/838,586
Granted
Sep 20, 2016
Kind
B2
Abstract

In a composition aspect of the invention, a nanoparticle coating comprises repeating polyacrylic acid monomers covalently bound together in an aliphatic chain having a plurality of carboxylic acid functional groups and modified carboxylic acid functional groups extending therefrom. A first portion of the modified carboxylic acid functional groups are modified by a PEG oligomer having a terminal methoxy functional group and a second portion of the modified carboxylic acid functional groups are modified by a PEG oligomer having at least one terminal sulfur moiety.

Claims (21)

1. A composition comprising:

nanoparticles surface-capped with a coating composition, the coating composition comprising:

repeating polyacrylic acid monomer units covalently bound together in an aliphatic chain having a plurality of carboxylic acid functional groups and modified carboxylic acid functional groups extending therefrom, wherein a first portion of the modified carboxylic acid functional groups are modified by a PEG oligomer having a terminal methoxy functional group and a second portion of the modified carboxylic acid functional groups are modified by a PEG oligomer having at least one terminal sulfur moiety.

2. The composition of claim 1 , wherein the nanoparticles are coated by being directly bound to the at least one terminal sulfur moiety.

3. The composition of claim 1 , wherein the nanoparticles are selected from metallic nanoparticles, semiconductor nanoparticles, or a combination thereof.

4. The composition of claim 1 , wherein the nanoparticles are selected from gold nanoparticles, ZnS nanoparticles, CdSe nanoparticles, or a combination thereof.

5. The composition of claim 1 , wherein the at least one terminal sulfur moiety is formed from thioctic acid.

6. The composition of claim 1 , wherein the at least one terminal sulfur moiety is formed from dihydrolipoic acid.

7. The composition of claim 1 , wherein the PEG oligomer having a terminal methoxy functional group is formed from a Compound 2 having a structure:

wherein n has a value such that an average molecular weight of the PEG oligomer is about 750.

8. The composition of claim 1 , wherein the PEG oligomer having at least one terminal sulfur moiety is formed from a Compound 1 having a structure:

wherein n has a value such that an average molecular weight of the PEG oligomer is about 600.

9. The composition of claim 1 , wherein the PEG oligomer having a terminal methoxy functional group is formed from a Compound 2 and the PEG oligomer having at least one terminal sulfur moiety is formed from a Compound 1; wherein the Compound 2 and the Compound 1 have the following structures:

wherein n has a value such that an average molecular weight of the PEG oligomer is about 750; and

wherein n has a value such that an average molecular weight of the PEG oligomer is about 600.

10. The composition of claim 1 , wherein the PEG oligomer having at least one terminal sulfur moiety is formed from dihydrolipoic acid.

11. The composition of claim 1 , further comprising a third portion of modified carboxylic acid functional groups, wherein the third portion of the modified carboxylic acid functional groups are modified by a PEG oligomer having a terminal azide functional group.

12. The composition of claim 11 , wherein the PEG oligomer having at least one terminal sulfur moiety is formed from a Compound 1 having a structure:

wherein n has a value such that an average molecular weight of the PEG oligomer is about 600.

13. The composition of claim 1 , wherein a third portion of the modified carboxylic acid functional groups are modified by a PEG oligomer having a terminal amine functional group.

14. The composition of claim 13 , wherein the PEG oligomer having at least one terminal sulfur moiety is formed from dihydrolipoic acid.

Assignments (2)
CONFIRMATORY LICENSE Recorded Apr 11, 2016
From: FLORIDA STATE UNIVERSITY
To: NATIONAL SCIENCE FOUNDATION
Reel/Frame 038401/0419 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Aug 28, 2015
From: MATTOUSSI, HEDI; PALUI, GOUTAM; NA, HYON BIN
To: THE FLORIDA STATE UNIVERSITY RESEARCH FOUNDATION, INC.
Reel/Frame 036446/0065 →
Continuity (4)
Division 13772595 · Feb 21, 2013
Continuation In Part 13608119 · Sep 10, 2012
Provisional Application 61532756 · Sep 9, 2011
Related Publication 20160136302A1 · May 19, 2016