IP Library Granted Patent US 9,486,453
Granted Patent B2
US 9,486,453 · App. 14/844,021 · Granted Nov 8, 2016

Composition and method for treatment of depression and psychosis in humans

Inventor: Daniel C. Javitt (Bardonia, NY)
Assignee: Glytech LLC
A61K31/496A61K31/06A61K31/135A61K31/138A61K31/381A61K31/42A61K31/431A61K31/4525A61K31/519A61K31/55A61K31/551A61K31/553A61K31/554A61K45/06
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Quick Facts
Patent No.
US 9,486,453
App. No.
14/844,021
Granted
Nov 8, 2016
Kind
B2
Abstract

Compositions and methods for the treatment of depression and psychoses in humans are disclosed. More particularly, the invention is directed to formulations containing antipsychotic and/or antidepressant medications and also containing an NMDAR antagonist. The present Invention Is also directed to methods tor the treatment of humans suffering from depression and other psychoses, including, schizophrenia, by administration of the inventive compositions in antidepressant and/or antipsychotic effective amounts.

Claims (12)

1. A method for reducing akathisia caused by lurasidone treatment in a subject with bipolar disorder, comprising:

administering an akathisia-inducing amount of lurasidone to the subject;

once akathisia is induced, continuing to administer lurasidone at a same dosage and frequency that caused akathisia; and

administering a therapeutically effective amount of a second composition comprising D-cycloserine (DCS) at a dosage in excess of 500 mg/day, wherein the DCS produces a NMDA receptor antagonistic blood plasma concentration measured at greater than 25 micrograms/mL,

thereby reducing akathisia.

2. A method for reducing the incidence of akathisia caused by lurasidone treatment in a subject with bipolar disorder, comprising:

administering therapeutically effective amounts of lurasidone, ketamine, and D-cycloserine (DCS) to a subject with bipolar disorder, wherein DCS is administered at a dosage in excess of 500 mg/day,

wherein the DCS produces a NMDA receptor antagonistic blood plasma concentration measured at greater than 25 micrograms/mL, thereby reducing the incidence of akathisia caused by lurasidone.

3. The method of claim 1 , wherein the lurasidone and second composition are administered intramuscularly, intravenously, intraperitoneally, parentally, or orally.

4. The method of claim 2 , wherein the lurasidone, ketamine, and D-cycloserine (DCS) are administered intramuscularly, intravenously, intraperitoneally, parentally, or orally.

5. The method of claim 1 , wherein the wherein the lurasidone and second composition are formulated as a single composition for administration to the subject.

6. The method of claim 2 , wherein the wherein the lurasidone, ketamine, and D-cycloserine (DCS) are formulated as a single composition for administration to the subject.

Assignments (2)
SECURITY INTEREST Recorded Sep 20, 2024
From: NRX PHARMACEUTICALS, INC.; HOPE THERAPEUTICS, INC.; NEURORX, INC.
To: ANSON INVESTMENTS MASTER FUND LP; ANSON EAST MASTER FUND LP
Reel/Frame 068647/0346 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Sep 3, 2015
From: JAVITT, DANIEL C.
To: GLYTECH, LLC
Reel/Frame 036539/0745 →
Continuity (4)
Division 13936198 · Jul 7, 2013
Provisional Application 61741114 · Jul 12, 2012
Provisional Application 61741115 · Jul 12, 2012
Related Publication 20150374684A1 · Dec 31, 2015