IP Library Granted Patent US 10,260,038
Granted Patent B2
US 10,260,038 · App. 14/890,296 · Granted Apr 16, 2019

Protein modification of living cells using sortase

Inventors: Lee Kim Swee (Heidelberg, DE); Hidde L. Ploegh (Brookline, MA)
Assignee: Whitehead Institute for Biomedical Research
C12N5/0006A61K39/0011A61K47/65A61K47/66A61K47/68C12N5/0636C12N5/0638C12N9/50A61K2039/5158C12Y304/2207
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Quick Facts
Patent No.
US 10,260,038
App. No.
14/890,296
Granted
Apr 16, 2019
Kind
B2
Abstract

Non-genetically engineered mammalian cells modified by sortase-mediated conjugation of an agent thereto are provided. Methods of conjugating agents to nongenetically engineered mammalian cells using sortase are provided. Methods of using the cells, e.g. a method of modulating an immune response of a subject to an entity of interest, a method of neutralizing a substance in the body of a subject, a method of treating a subject in need of treatment for deficiency of a protein, and a method of treating a subject in need of treatment for a disease, are provided.

Claims (17)

1. A human cell having a binding moiety or therapeutic agent linked thereto via a sortase recognition sequence, wherein the binding moiety or therapeutic agent is linked to an endogenous, non-genetically engineered protein expressed by the human cell, and wherein the human cell has not been genetically engineered to express a polypeptide comprising a sortase recognition sequence, wherein the binding moiety or therapeutic agent comprises an immune checkpoint inhibitor.

2. The human cell of claim 1 , wherein the human cell is an immune system cell.

3. The human cell of claim 1 , wherein the sortase recognition sequence comprises LPXTG.

4. The human cell of claim 1 , wherein the binding moiety comprises a targeting moiety that binds to an epitope or antigen of interest.

5. The human cell of claim 1 , wherein the binding moiety comprises a monoclonal antibody, a single chain antibody, or a single domain antibody.

6. The human cell of claim 5 , wherein the binding moiety comprises a VHH.

7. The human cell of claim 1 , wherein the human cell is selected from the group consisting of a red blood cell, a peripheral blood mononuclear cell, a lymphocyte, a T cell, a NK cell, and a dendritic cell.

8. The human cell of claim 1 , wherein the human cell is a non-immortalized cell.

9. The human cell of claim 1 , wherein the human cell is a primary cell.

10. The human cell of claim 1 , wherein the human cell has not been genetically engineered to express a polypeptide comprising a sequence comprising one or more N-terminal glycines.

11. The human cell of claim 1 , wherein the human cell has not been genetically engineered.

12. A method of treating a subject in need of treatment for a disease, the method comprising administering at least one human cell of claim 1 to the subject, wherein the at least one cell is effective for treating the disease.

13. The method of claim 12 , wherein the human cell originates from the subject and said subject is in need of evaluation or treatment for a disease of interest or from a donor who is immunocompatible with the subject.

14. The method of claim 13 , wherein the human cell originates from the subject in need of evaluation or treatment for a disease characterized by the presence of abnormal or excessive cells or pathogens in the subject's body, or from a donor who is immunocompatible with the subject.

15. The method of claim 14 , wherein the human cell originates from the subject in need of evaluation or treatment for cancer, an autoimmune disease, or an infection or from a donor who is immunocompatible with the subject.

16. A mammalian cell having a binding moiety or therapeutic agent linked thereto via a sortase recognition sequence, wherein the binding moiety or therapeutic agent is linked to an endogenous, non-genetically engineered protein expressed by the mammalian cell, and wherein the binding moiety or therapeutic agent comprises an immune checkpoint inhibitor.

17. A method of treating a subject in need of treatment for a disease, the method comprising administering the mammalian cell of claim 16 to the subject.

Assignments (2)
CONFIRMATORY LICENSE Recorded Aug 7, 2017
From: WHITEHEAD INSTITUTE FOR BIOMEDICAL RES
To: NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT
Reel/Frame 043458/0054 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Nov 19, 2015
From: PLOEGH, HIDDE L.; SWEE, LEE KIM
To: WHITEHEAD INSTITUTE FOR BIOMEDICAL RESEARCH
Reel/Frame 037087/0761 →
Continuity (3)
Provisional Application 61943094 · Feb 21, 2014
Provisional Application 61822092 · May 10, 2013
Related Publication 20160122707A1 · May 5, 2016
Cited By (3)
US 50,550 US 12,331,311 US 12,656,341