IP Library Granted Patent US 9,827,222
Granted Patent B2
US 9,827,222 · App. 14/901,976 · Granted Nov 28, 2017

Treating or preventing nephrogenic diabetes insipidus

Inventors: Jeff M. Sands (Atlanta, GA); Mitsi A. Blount (Atlanta, GA); Janet D. Klein (Decatur, GA)
Assignee: Emory University
A61K31/343A61K31/155A61K31/341A61K31/405A61K31/427A61K31/4365A61K31/4965A61K31/549A61K31/7056A61K31/7076A61K33/00A61K45/06
View Patent ↗
Loading inventors, assignments & file history…
Monitor This Case
Get email alerts when status or documents change.
Order Certified Copies
Most orders are placed with the USPTO same day — all within 24 business hours.
Order via The Patent Place →
Pre-filled with this patent's details
Quick Facts
Patent No.
US 9,827,222
App. No.
14/901,976
Granted
Nov 28, 2017
Kind
B2
Abstract

In certain embodiments, the disclosure relates to methods of treating or preventing nephrogenic diabetes insipidus comprising administering an effective amount of a AMPK activator to a subject in need thereof, wherein In certain embodiments, the AMPK activator is metformin or salt thereof. In certain embodiments, the subject has been diagnosed with nephrogenic diabetes insipidus.

Claims (9)

1. A method of treating nephrogenic diabetes insipidus comprising administering an effective amount of an AMPK activator to a subject in need thereof wherein the subject has symptoms of excessive urination and excessive thirst wherein urine of the subject does not contain glucose.

2. The method of claim 1 , wherein the AMPK activator is metformin or salt thereof.

3. The method of claim 1 , wherein the subject has been diagnosed with nephrogenic diabetes insipidus.

4. The method of claim 1 , wherein the subject is restricted from drinking water and an hourly increase in osmolality of urine of the subject is less than 30 mOsm/kg per hour for at least 3 hours.

5. The method of claim 1 , wherein the subject is not responsive to vasopressin.

6. The method of claim 1 , wherein the AMPK activator is administered in combination with a thiazide, indomethacin, amiloride, or other diuretic.

7. The method of claim 1 , wherein the AMPK activator is administered in combination with lithium.

8. The method of claim 1 , wherein the AMPK activator is cryptotanshinone.

9. The method of claim 1 , wherein the AMPK activator is 5-aminoimidazole-4-carboxamide-1-beta-D-ribofuranoside, A-769662 [4-hydroxy-3-(2′-hydroxy-[1,1′-biphenyl]-4-yl)-6-oxo-6,7-dihydrothieno[2,3-b]pyridine-5-carbonitrile], D942 [5-(3-(4-(2-(4-Fluorophenyl) ethoxy)phenyl)propyl)furan-2-carboxylic acid], WS070117 [O2′,O3′,O5′-tri-acetyl-N6-(3-hydroxylaniline)adenosine], PT1 [2-Chloro-5-[[5-[[5-(4,5-Dimethyl-2-nitrophenyl)-2-furanyl]methylene]-4,5-dihydro-4-ox-o-2-thiazolyl]amino]benzoic acid] or salts thereof.

Assignments (1)
CONFIRMATORY LICENSE Recorded Jun 13, 2016
From: EMORY UNIVERSITY
To: NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT
Reel/Frame 038964/0695 →
Continuity (2)
Provisional Application 61841648 · Jul 1, 2013
Related Publication 20160367516A1 · Dec 22, 2016