IP Library Granted Patent US 9,517,238
Granted Patent B2
US 9,517,238 · App. 14/934,589 · Granted Dec 13, 2016

Compositions and methods for treating allergic inflammation through inhibition of NTRK1

Inventors: Mark Rochman (Cincinnati, OH); Marc E. Rothenberg (Cincinnati, OH)
Assignee: CHILDREN'S HOSPITAL MEDICAL CENTER
A61K31/553A61K31/00A61K31/4545A61K45/06
View Patent ↗
Loading inventors, assignments & file history…
Monitor This Case
Get email alerts when status or documents change.
Order Certified Copies
Most orders are placed with the USPTO same day — all within 24 business hours.
Order via The Patent Place →
Pre-filled with this patent's details
Quick Facts
Patent No.
US 9,517,238
App. No.
14/934,589
Granted
Dec 13, 2016
Kind
B2
Abstract

The invention provides methods of treating allergic inflammatory conditions using an anti-neurotrophin tyrosine kinase receptor 1 (NTRK1)-based therapeutic agent, and related compositions and methods.

Claims (10)

1. A method of treating eosinophilic esophagitis (EoE) in a human subject in need thereof, comprising administering to the subject an amount of a tyrosine kinase inhibitor effective to suppress NTRK1 activity in target cells of the human subject, wherein the tyrosine kinase inhibitor is lestaurtinib (CEP-701) or crizotinib.

2. The method of claim 1 , wherein the target cells are epithelial cells.

3. The method of claim 1 , wherein the target cells are cells of a target tissue in the subject.

4. The method of claim 1 , wherein the target tissue is tracheal, lung, or esophageal tissue.

5. The method of claim 1 , wherein the tyrosine kinase inhibitor is effective to suppress NTRK1 activity in the cells of the subject, relative to untreated cells.

6. The method of claim 5 , wherein the tyrosine kinase inhibitor is effective to suppress NTRK1 gene expression or protein expression, or both.

7. The method of claim 1 , wherein the amount of the tyrosine kinase inhibitor is effective to ameliorate one or more symptoms of the EoE.

8. The method of claim 1 , further comprising administering to the subject at least one additional active agent.

9. The method of claim 8 , wherein the at least one additional active agent is an anti-inflammatory agent.

10. The method of claim 8 , wherein the at least one additional active agent is an IL-13 inhibitor, a non-steroidal anti-inflammatory drug (NSAID), a cytokine inhibitor, or a steroid.

Assignments (2)
CONFIRMATORY LICENSE Recorded Dec 1, 2016
From: CINCINNATI CHILDRENS HOSP MED CTR
To: NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT
Reel/Frame 040787/0680 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Nov 19, 2015
From: ROTHENBERG, MARC E; ROCHMAN, MARK
To: CHILDREN'S HOSPITAL MEDICAL CENTER
Reel/Frame 037084/0278 →
Continuity (2)
Provisional Application 62076719 · Nov 7, 2014
Related Publication 20160129012A1 · May 12, 2016