IP Library › Granted Patent US 10,023,891
Granted Patent B2
US 10,023,891 · App. 15/033,570 · Granted Jul 17, 2018

Process of chiral resolution of cyclic and acyclic acetates to enantiomerically pure (R)-alcohols

Inventors: Dipesh Dattu Jadhav (Maharashtra, IN); Nilofer Jahan Khairunnasar Siddiqui (Maharashtra, IN); Swati Pramod Kolet (Maharashtra, IN); Hirekodathakallu Thulasiram (Maharashtra, IN)
Assignee: COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH
C12P17/182C12P7/02C12P7/04C12P7/22C12P7/26C12P41/004
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Quick Facts
Patent No.
US 10,023,891
App. No.
15/033,570
Granted
Jul 17, 2018
Kind
B2
Abstract

The patent discloses herein a process for the chiral resolution of racemic cyclic and acyclic acetates to obtain (R)-alcohol. Further, it discloses the resolution of racemic cyclic and acyclic acetates to obtain enantiomerically pure (R)-(−)-alcohol as single enantiomer through fungal catalyzed deacylation in single fermentation, wherein fungal strains are F. proliferatum.

Claims (8)

1. A process for chiral resolution of a racemic acetate to obtain an enantiomerically pure (R)-Alcohol as a single enantiomer comprising the steps of:

i) incubating Fusarium proliferatum for from 24 to 48 hours at a temperature between 28° C. to 30° C. in a medium;

ii) adding the racemic acetate to the medium after step i) and incubating further for from 6 hours to 3 days at temperature between 28° C. to 30° C. to obtain the enantiomerically pure (R)-Alcohol.

2. The process according to claim 1 , wherein the Fusarium proliferatum comprises spores and mycelia.

3. The process according to claim 1 , wherein the racemic acetate is selected from the group consisting of 2-Heptyl acetate, lavandulyl acetate and 2-Hexyl acetate.

4. The process according to claim 1 , wherein the racemic acetate is a cyclic racemic acetate or an acyclic racemic acetate.

5. The process according to claim 1 , wherein a yield of the enantiomerically pure (R)-Alcohol as a single enantiomer is 95-99.9%.

6. The process according to claim 1 , wherein the enantiomerically pure (R)-Alcohol is selected from the group consisting of R-lavandulol, R-2-Hexnol, R-2-Heptanol, R-1-Phenyl ethanol and R-1-Phenyl propanol.

Assignments (1)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Sep 1, 2016
From: JADHAV, DIPESH DATTU; SIDDIQUI, NILOFER JAHAN; KOLET, SWATI PRAMOD; THULASIRAM, HIREKODATHAKALLU
To: COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH
Reel/Frame 039617/0355 →
Priority Claims (1)
IN 3242/DEL/2013 · Nov 1, 2013 · national
Continuity (1)
Related Publication 20160281122A1 · Sep 29, 2016