IP Library Granted Patent US 11,446,309
Granted Patent B2
US 11,446,309 · App. 15/034,922 · Granted Sep 20, 2022

Combination therapy for cancer using bromodomain and extra-terminal (BET) protein inhibitors

Inventors: James E. Bradner (Weston, MA); Michael R. McKeown (Brookline, MA); Margaret A. Shipp (Wellesley, MA); Bjoern Chapuy (Boston, MA); Kwok-kin Wong (Arlington, MA); Zhao Chen (Sharon, MA)
Assignee: Dana-Farber Cancer Institute, Inc.
A61K31/551A61K31/404A61K31/453A61K31/5377A61K45/06A61P35/00C07D487/04C07D495/14
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Quick Facts
Patent No.
US 11,446,309
App. No.
15/034,922
Granted
Sep 20, 2022
Kind
B2
Abstract

The present invention provides methods for treating cancer using combinations of bromodomain and extra-terminal (BET) protein inhibitors and certain chemotherapeutic drugs.

Claims (10)

1. A method of treating diffuse large B-cell lymphoma (DLBCL) comprising:

administering to a subject in need thereof a first agent, S-JQ35:

or a pharmaceutically acceptable salt thereof,

in combination with one or more second agents selected from ABT263, or ABT199,

wherein the first agent and the one or more second agents are administered in an amount effective to treat the DLBCL.

2. The method of claim 1 , wherein the first agent and the one or more second agents are administered sequentially or simultaneously.

3. The method of claim 1 , wherein the subject is a mammal.

4. The method claim 3 , wherein the subject is a human patient.

5. The method of claim 1 , further comprising treating the subject with an additional anti-neoplasia therapy.

6. The method of claim 5 , wherein the additional anti-neoplasia therapy is surgery, radiation therapy, chemotherapy, gene therapy, DNA therapy, viral therapy, RNA therapy, adjuvant therapy, immunotherapy or a combination thereof.

Assignments (2)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Sep 24, 2018
From: BRADNER, JAMES E.; MCKEOWN, MICHAEL R.; SHIPP, MARGARET A.; CHAPUY, BJOERN; WONG, KWOK KIN; CHEN, ZHAO
To: DANA-FARBER CANCER INSTITUTE, INC.
Reel/Frame 047130/0079 →
CONFIRMATORY LICENSE Recorded Jul 1, 2016
From: DANA-FARBER CANCER INST
To: NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT
Reel/Frame 039237/0064 →
Continuity (2)
Provisional Application 61901908 · Nov 8, 2013
Related Publication 20160279141A1 · Sep 29, 2016