IP Library Granted Patent US 9,610,279
Granted Patent B2
US 9,610,279 · App. 15/080,899 · Granted Apr 4, 2017

Method for induction of a heat shock protein, anti-stress or regulation of an autonomic nerve

Inventors: Hiroshi Nishioka (Hokkaido, JP); Tomohiro Ito (Hokkaido, JP); Takahiro Maeda (Hokkaido, JP)
Assignee: AMINO UP CHEMICAL CO., LTD.
A61K31/4025A23L19/09A23L33/105A61K31/341A61K36/8965C07D307/48C07D307/50C07D405/12A61K2236/37A61K2236/39
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Quick Facts
Patent No.
US 9,610,279
App. No.
15/080,899
Granted
Apr 4, 2017
Kind
B2
Abstract

A method for induction of a heat shock protein, anti-stress or regulation of an autonomic nerve comprises: administering a mammalian subject in need thereof a composition comprising an effective amount of hydroxymethylfurfural derivative of the following formula: wherein R is selected from the group consisting of formula (I): (II): HOOCCH 2 COCO—, (III): HOOCCH 2 CH 2 COCO—, and (IV): a hydrogen atom.

Claims (27)

1. A method for induction of a heat shock protein, anti-stress, or regulation of an autonomic nerve comprising administering a mammalian subject in need thereof once or twice daily a composition comprising an effective amount of hydroxymethylfurfural derivative of the following formula:

wherein R is selected from the group consisting of formula (I):

(II): HOOCCH 2 COCO—, and (III): HOOCCH 2 CH 2 COCO—, at a dosage of 50 mg to 2000 mg per day, wherein the dosage is in a form selected from the group consisting of granules, particulates, tablets, capsules, suspensions, aqueous solutions, emulsions, and powders.

2. The method according to claim 1 wherein the hydroxymethylfurfural derivative is obtained by heat-treating an asparagus stem with hot water and an enzyme treatment,

wherein the enzyme treatment is carried out by adding at least one enzyme selected from among a group consisting of cellulase, hemicellulase, pectinase, amylase and pullulanase; and treating at a temperature of 30 to 60° C., for 1 to 72 hours.

3. The method of claim 1 wherein the composition comprises powders prepared by a method comprising: heat-treating an asparagus stem with hot water to obtain a heat-treated mixture for about 20 to 180 minutes; cooling; filtering; concentrating; adding a pharmaceutically acceptable excipient; and drying.

4. The method of claim 1 wherein the dosage is in a form selected from the group consisting of tablets, capsules, suspensions, aqueous solutions, emulsions, and powders.

5. A method for induction of a heat shock protein, anti-stress, or regulation of an autonomic nerve comprising:

heat-treating an asparagus stem with hot water and an enzyme treatment, wherein the enzyme treatment is carried out by adding at least one enzyme selected from the group consisting of cellulase, hemicellulase, pectinase, amylase, and pullulanase, at a temperature of 30° C. to 60° C. for 1 to 72 hours,

administering the resulting product to a mammalian subject in need thereof, and

evaluating heat shock protein activity, stress, autonomic nervous balance, or autonomic nervous activity of the mammalian subject.

6. The method of claim 5 wherein the product is in a form selected from the group consisting of granules, particulates, tablets, capsules, suspensions, aqueous solutions, emulsions, and powders, and administered once or twice daily at a dosage of 50 mg to 2000 mg per day.

7. The method of claim 6 wherein the product is in a form selected from the group consisting of tablets, capsules, suspensions, aqueous solutions, emulsions, and powders.

8. A method for induction of a heat shock protein, anti-stress or regulation of an autonomic nerve comprising:

administering a mammalian subject in need thereof a composition comprising an effective amount of hydroxymethylfurfural derivative of the following formula:

wherein R is selected from the group consisting of formula (I):

(II): HOOCCH 2 COCO—, and (III): HOOCCH 2 CH 2 COCO—, and

evaluating heat shock protein activity, stress, autonomic nervous balance, or autonomic nervous activity of the mammalian subject.

9. The method of claim 8 wherein the evaluating step is conducted at least once before the administrating step and at least once after the administrating step.

10. The method of claim 8 wherein the administrating step comprises administrating the mammalian subject the composition 50 mg to 2000 mg/day.

11. The method of claim 8 wherein the administrating step comprises administrating the mammalian subject the composition once or twice daily.

12. The method of claim 8 wherein the composition is in a dosage form selected from the group consisting of granules, particulates, tablets, capsules, suspensions, aqueous solutions, emulsions, and powders.

13. The method according to claim 8 wherein the composition is in a dosage form selected from the group consisting of tablets, capsules, suspensions, aqueous solutions, emulsions, and powders.

14. The method according to claim 8 wherein the hydroxymethylfurfural derivative is obtained by heat-treating an asparagus stem with hot water and an enzyme treatment,

wherein the enzyme treatment is carried out by adding at least one enzyme selected from among a group consisting of cellulase, hemicellulase, pectinase, amylase and pullulanase; and

treating at a temperature of 30 to 60° C., for 1 to 72 hours.

15. The method of claim 8 wherein the composition comprises powders prepared by a method comprising: heat-treating an asparagus stem with hot water to obtain a heat-treated mixture for about 20 to 180 minutes; cooling; filtering; concentrating; adding an pharmaceutically acceptable excipient; and drying.

Assignments (2)
CHANGE OF NAME Recorded Jul 9, 2019
From: AMINO UP CHEMICAL CO., LTD.
To: AMINO UP CO., LTD.
Reel/Frame 049707/0144 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Mar 25, 2016
From: NISHIOKA, HIROSHI; ITO, TOMOHIRO; MAEDA, TAKAHIRO
To: AMINO UP CHEMICAL CO., LTD.
Reel/Frame 038100/0812 →
Priority Claims (1)
JP 2011-277926 · Dec 20, 2011 · national
Continuity (2)
Continuation 14366276
Related Publication 20160193184A1 · Jul 7, 2016