IP Library › Patent Application 15094777
Patent Application
App. No. 15/094,777

MACROCYCLIC INHIBITORS OF FLAVIVIRIDAE VIRUSES

Loading inventors, assignments & file history…
Monitor This Case
Get email alerts when status or documents change.
Order Certified Copies
Most orders are placed with the USPTO same day — all within 24 business hours.
Order via The Patent Place →
Pre-filled with this patent's details
Quick Facts
Patent No.
US None
App. No.
15/094,777
Abstract

Provided are compounds of Formula I: and pharmaceutically acceptable salts and esters thereof. The compounds, compositions, and methods provided are useful for the treatment of virus infections, particularly hepatitis C infections.

Claims (8)

1 - 37 . (canceled)

38 . A method of treating a Flaviviridae viral infection in a human patient in need thereof, comprising administering to the patient a therapeutically effective amount of a compound selected from the group consisting of:

or a pharmaceutically acceptable salt, isotope, stereoisomer, mixture of stereoisomers, tautomer, ester or prodrug thereof.

39 . A method according to claim 38 wherein the compound is

or a pharmaceutically acceptable salt, isotope, stereoisomer, mixture of stereoisomers, tautomer, ester or prodrug thereof.

40 . A method according to claim 38 wherein the compound is

41 . A method according to claim 38 wherein the Flaviviridae infection is caused by a virus selected from the group consisting of West Nile virus (WNV) Japanese encephalitis virus (JEV), tick-borne encephalitis virus, Junjin virus, Murray Valley encephalitis, St Louis enchaplitis, Omsk hemorrhagic fever virus and Zika virus.

42 . A method according to claim 38 wherein the Flaviviridae infection is caused by Zika virus.

Assignments (2)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jun 23, 2017
From: SELCIA LIMITED
To: CYPRALIS LIMITED
Reel/Frame 042800/0596 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded May 12, 2016
From: STEADMAN, VICTORIA ALEXANDRA; POULLENNEC, KARINE G.; LAZARIDES, LINOS; ACIRO, CAROLINE; DEAN, DAVID KENNETH; KEATS, ANDREW JOHN; SIEGEL, DUSTIN SCOTT; SCHRIER, ADAM JAMES; MACKMAN, RICHARD; JANSA, PETR; WATT, GREG; HIGHTON, ADRIAN JOHN; CHIVA, JEAN YVES
To: GILEAD SCIENCES, INC.; SELCIA LTD.
Reel/Frame 038569/0338 →