IP Library Granted Patent US 9,770,482
Granted Patent B2
US 9,770,482 · App. 15/139,066 · Granted Sep 26, 2017

Targeting the EGFR-SGLT1 interaction for cancer therapy

Inventor: Zhang Weihua (Houston, TX)
Assignee: The University of Houston System
A61K38/10A61K31/422A61K31/517A61K31/519A61K31/5377A61K31/70A61K31/7034A61K31/7042A61K38/179A61K45/06C07K7/08
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Quick Facts
Patent No.
US 9,770,482
App. No.
15/139,066
Granted
Sep 26, 2017
Kind
B2
Abstract

A compound can destabilize an epidermal growth factor receptor (EGFR) protein and a sodium/glucose co-transporter 1 (SGLT 1) protein. In one embodiment, the compound is a peptide derived from the interacting domain of EGFR. In another embodiment, the peptide is administered to a patient to treat cancer.

Claims (8)

1. A method of treating cancer cells comprising:

identifying a subject having cancer cells that express an epidermal growth factor receptor (EGFR) protein and a sodium/glucose co-transporter 1 (SGLT1) protein;

treating the cancer cells by administering to the subject a peptide capable of destabilizing both EGFR and SGLT1 proteins, wherein the peptide consists of one of SEQ ID NO: 001, SEQ ID NO: 002, SEQ ID NO: 003, SEQ ID NO: 004, SEQ ID NO: 005, SEQ ID NO: 006, SEQ ID NO: 007, SEQ ID NO: 008, SEQ ID NO: 009, SEQ ID NO: 010, and SEQ ID NO: 011.

2. The method of claim 1 , further comprising co-administering to the subject a tyrosine-kinase inhibitor with the peptide.

3. The method of claim 1 , wherein the peptide is administered to cause the death of cancer cells.

4. The method of claim 1 , wherein the cancer cells include at least one of breast cancer cells, prostate cancer cells, and colon cancer cells.

5. The method of claim 2 , wherein the tyrosine-kinase inhibitor is at least one of Gefitnib, Erlotinib, Icontinib, Mubritinib, Vandertanib, Lapatinib, Peletinib, Canetinib, Neratinib, Afatinib, and Dacomitinib.

6. The method of claim 1 , wherein the cancer cells are at least one of breast cancer cells, prostate cancer cells, colon cancer cells, ovarian cancer cells, oral squamous cancer cells, and pancreatic cancer cells.

Assignments (2)
CONFIRMATORY LICENSE Recorded Jun 22, 2023
From: UNIVERSITY OF HOUSTON
To: UNITED STATES GOVERNMENT
Reel/Frame 064067/0123 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Apr 26, 2016
From: WEIHUA, ZHANG
To: THE UNIVERSITY OF HOUSTON SYSTEM
Reel/Frame 038387/0528 →
Continuity (3)
Division 14273375 · May 8, 2014
Provisional Application 61821028 · May 8, 2013
Related Publication 20160228495A1 · Aug 11, 2016