IP Library Granted Patent US 10,017,575
Granted Patent B2
US 10,017,575 · App. 15/242,135 · Granted Jul 10, 2018

Antibody molecules having specificity for human OX40

Inventors: Alastair David Griffiths Lawson (Slough, GB); Andrew Malcolm Nesbitt (Slough, GB); Andrew George Popplewell (Slough, GB); Stevan Graham Shaw (Slough, GB); Diana Shpektor (Shoreline, WA); Yi Zhang (San Francisco, CA)
Assignee: UCB Pharma S.A.
C07K16/2878A61K39/3955A61K45/06C07K14/70578A61K2039/505C07K2317/24C07K2317/33C07K2317/55C07K2317/565C07K2317/73C07K2317/76C07K2317/92
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Quick Facts
Patent No.
US 10,017,575
App. No.
15/242,135
Granted
Jul 10, 2018
Kind
B2
Abstract

The invention relates to antibody molecules having specificity for antigenic determinants of human OX40, therapeutic uses of the antibody molecules and methods for producing said antibody molecules.

Claims (53)

1. An antibody that binds human OX40 comprising a light chain comprising a variable domain that comprises a sequence having at least 95% identity to the sequence given in SEQ ID NO:9and a heavy chain comprising a variable domain that comprises a sequence having at least 95% identity to the sequence given in SEQ ID NO:7.

2. The antibody of claim 1 , wherein the light chain comprises a variable domain that comprises a sequence having at least 98% identity to the sequence given in SEQ ID NO:9.

3. The antibody of claim 1 , wherein the light chain comprises a light chain comprising a variable domain that comprises the sequence given in SEQ ID NO:9.

4. The antibody of claim 1 , wherein the light chain comprises a heavy chain comprising a variable domain that comprises a sequence having at least 98% identity to the sequence given in SEQ ID NO:7.

5. The antibody of claim 1 , wherein the light chain comprises a heavy chain comprising a variable domain that comprises the sequence given in SEQ ID NO:7.

6. An antibody that binds human OX40, comprising a heavy chain that comprises a sequence that has at least 95% identity to the sequence given in SEQ ID NO:15 and a light chain that comprises a sequence that has at least 95% identity to the sequence given in SEQ ID NO:11.

7. The antibody of claim 6 , wherein the heavy chain comprises a sequence having at least 98% identity to the sequence given in SEQ ID NO:15.

8. The antibody of claim 6 , wherein the heavy chain comprises the sequence given in SEQ ID NO:15.

9. The antibody of claim 6 , wherein the light chain comprises a sequence having at least 98% identity to the sequence given in SEQ ID NO:11.

10. The antibody of claim 6 , wherein the light chain comprises the sequence given in SEQ ID NO:11.

11. The antibody of claim 1 , wherein the antibody is a complete antibody molecule having full length heavy and light chains.

12. The antibody of claim 1 , wherein the antibody is a fragment of a complete antibody molecule.

13. The antibody of claim 6 , wherein the antibody is a complete antibody molecule having full length heavy and light chains.

14. The antibody of claim 6 , wherein the antibody is a fragment of a complete antibody molecule.

15. An antibody heavy chain comprising the sequence given in SEQ ID NO:1 for CDR-H1, the sequence given in SEQ ID NO:2 or SEQ ID NO:20 for CDR-H2 and the sequence given in SEQ ID NO:3 for CDR-H3.

16. An antibody light chain comprising the sequence given in SEQ ID NO:4 or SEQ ID NO:21 for CDR-L1, a CDR having the sequence given in SEQ ID NO:5 for CDR-L2 and a CDR having the sequence given in SEQ ID NO:6 for CDR-L3.

17. A fusion protein comprising:

an OX40-binding immunoglobulin; and

two single domain antibodies linked to the OX40-binding immunoglobulin;

wherein the OX40-binding immunoglobulin comprises a heavy chain and a light chain, wherein:

the heavy chain comprises a variable domain that comprises the sequence given in SEQ ID NO:1 for CDR-H1, a CDR having the sequence given in SEQ ID NO:2 or SEQ ID NO:20 for CDR-H2 and a CDR having the sequence given in SEQ ID NO:3 for CDR-H3; and

the light chain comprises variable domain that comprises the sequence given in SEQ ID NO:4 or SEQ ID NO:21 for CDR-L1, a CDR having the sequence given in SEQ ID NO:5 for CDR-L2 and a CDR having the sequence given in SEQ ID NO:6 for CDR-L3; or

the heavy chain comprises a variable domain that comprises a sequence having at least 95% identity to the sequence given in SEQ ID NO:7; and

the light chain comprises a variable domain that comprises a sequence having at least 95% identity to the sequence given in SEQ ID NO:9.

18. The fusion protein of claim 17 , wherein:

the heavy chain comprises a variable domain that comprises the sequence given in SEQ ID NO:1 for CDR-H1, a CDR having the sequence given in SEQ ID NO:2 or SEQ ID NO:20 for CDR-H2 and a CDR having the sequence given in SEQ ID NO:3 for CDR-H3; and

the light chain comprises variable domain that comprises the sequence given in SEQ ID NO:4 or SEQ ID NO:21 for CDR-L1, a CDR having the sequence given in SEQ ID NO:5 for CDR-L2 and a CDR having the sequence given in SEQ ID NO:6 for CDR-L3.

19. The fusion protein of claim 17 , wherein:

the heavy chain comprises a variable domain that comprises a sequence having at least 95% identity to the sequence given in SEQ ID NO:7; and

the light chain comprises a variable domain that comprises a sequence having at least 95% identity to the sequence given in SEQ ID NO:9.

20. The fusion protein of claim 19 , wherein:

the heavy chain comprises a variable domain that comprises a sequence having at least 98% identity to the sequence given in SEQ ID NO:7; and

the light chain comprises a variable domain that comprises a sequence having at least 98% identity to the sequence given in SEQ ID NO:9.

21. The fusion protein of claim 20 , wherein:

the heavy chain comprises a variable domain that comprises the sequence given in SEQ ID NO:7; and

the light chain comprises a variable domain that comprises the sequence given in SEQ ID NO:9.

22. The fusion protein of claim 17 , wherein the immunoglobulin is a Fab or Fab' fragment.

23. The fusion protein of claim 17 , wherein the two single domain antibodies are a variable heavy (VH) and variable light (VL) pairing.

24. The fusion protein of claim 23 , wherein the two single domain antibodies are linked by a disulfide bond.

25. The fusion protein of claim 23 , wherein the variable heavy (VH) and variable light (VL) pairing provides an albumin binding site.

26. The fusion protein of claim 17 , wherein

the heavy chain comprises a variable domain that comprises the sequence given in SEQ ID NO:1 for CDR-H1, a CDR having the sequence given in SEQ ID NO:2 or SEQ ID NO:20 for CDR-H2 and a CDR having the sequence given in SEQ ID NO:3 for CDR-H3; and

the light chain comprises variable domain that comprises the sequence given in SEQ ID NO:4 or SEQ ID NO:21 for CDR-L1, a CDR having the sequence given in SEQ ID NO:5 for CDR-L2 and a CDR having the sequence given in SEQ ID NO:6 for CDR-L3; and

the two single domain antibodies are a variable heavy (VH) and variable light (VL) pairing that provides an albumin binding site.

27. The fusion protein of claim 26 , wherein the two single domain antibodies are linked by a disulfide bond.

28. The fusion protein of claim 17 , wherein

the heavy chain comprises a variable domain that comprises the sequence given in SEQ ID NO:1 for CDR-H1, a CDR having the sequence given in SEQ ID NO:2 or SEQ ID NO:20 for CDR-H2 and a CDR having the sequence given in SEQ ID NO:3 for CDR-H3; and

the light chain comprises variable domain that comprises the sequence given in SEQ ID NO:4 or SEQ ID NO:21 for CDR-L1, a CDR having the sequence given in SEQ ID NO:5 for CDR-L2and a CDR having the sequence given in SEQ ID NO:6 for CDR-L3; and

the two single domain antibodies are a variable heavy (VH) and variable light (VL) pairing that provides an albumin binding site.

29. The fusion protein of claim 28 , wherein the two single domain antibodies are linked by a disulfide bond.

30. An antibody comprising a heavy chain according to claim 15 .

31. An antibody heavy chain comprising the sequence given in SEQ ID NO:3 for CDR-H3.

32. An antibody comprising a heavy chain according to claim 31 .

Assignments (2)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Dec 18, 2017
From: UCB PHARMA S.A.
To: UCB BIOPHARMA SPRL
Reel/Frame 044418/0768 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Aug 22, 2016
From: GRIFFITHS LAWSON, ALASTAIR DAVID; NESBITT, ANDREW MALCOLM; POPPLEWELL, ANDREW GEORGE; SHAW, STEVAN GRAHAM; SHPEKTOR, DIANA; ZHANG, YI
To: UCB PHARMA S.A.
Reel/Frame 039499/0591 →
Continuity (4)
Division 13973189 · Aug 22, 2013
Division 12706993 · Feb 17, 2010
Provisional Application 61153038 · Feb 17, 2009
Related Publication 20160355598A1 · Dec 8, 2016
Cited By (1)
US 12,742,015