IP Library Granted Patent US 10,105,415
Granted Patent B2
US 10,105,415 · App. 15/328,426 · Granted Oct 23, 2018

Compositions comprising granulocyte-macrophage colony-stimulating factor for the treatment of inflammatory bowel disease

Inventors: Lars Heslet (Gentofte, DK); Lars Otto Uttenthal (Salamanca, ES)
Assignee: Reponex Pharmaceuticals A/S
A61K38/193A61K9/0031A61K9/08A61K9/1075A61K9/127A61K31/4164A61K31/665A61K35/741A61K45/06
View Patent ↗
Loading inventors, assignments & file history…
Monitor This Case
Get email alerts when status or documents change.
Order Certified Copies
Most orders are placed with the USPTO same day — all within 24 business hours.
Order via The Patent Place →
Pre-filled with this patent's details
Quick Facts
Patent No.
US 10,105,415
App. No.
15/328,426
Granted
Oct 23, 2018
Kind
B2
Abstract

The present invention provides compositions comprising granulocyte-macrophage colony-stimulating factor and fosfomycin for the treatment, prevention or alleviation of an inflammatory bowel disease such as Crohn's disease, ulcerative colitis or necrotizing enterocolitis of newborn and premature infants by administration of the compositions into the intestinal lumen.

Claims (12)

1. A method of alleviating the symptoms of inflammatory bowel disease, comprising:

selecting a patient that has inflammatory bowel disease;

administering to said selected patient locally into a bowel lumen an effective amount of a composition comprising a granulocyte-macrophage colony-stimulating factor (GM-CSF), molgramostim or sargramostim, fosfomycin and metronidazole.

2. The method of alleviating the symptoms of the inflammatory bowel disease according to claim 1 , wherein said inflammatory bowel disease is any one of Crohn's disease, ulcerative colitis or necrotizing enterocolitis.

3. The method of alleviating the symptoms of the inflammatory bowel disease according to claim 2 , wherein said inflammatory bowel disease is ulcerative colitis and wherein the composition is for local administration into the lumen of an affected area of any one of the ascending, transverse, descending and sigmoid colon or rectum.

4. The method of alleviating the symptoms of the inflammatory bowel disease according to claim 2 , wherein said inflammatory bowel disease is necrotizing enterocolitis in a newborn or premature infant and wherein the composition is for local administration into the lumen of an affected area of any one of the ascending, transverse, descending and sigmoid colon or rectum.

5. The method of alleviating the symptoms of the inflammatory bowel disease according to claim 4 , wherein the GM-CSF is in a formulation comprising liposome or micelle or microcapsule or nanoparticle.

6. The method of alleviating the symptoms of the inflammatory bowel disease according to claim 5 , wherein the composition further comprises one or more protease inhibitors suitable for in-vivo administration into the bowel lumen.

7. The method of alleviating the symptoms of the inflammatory bowel disease according to claim 6 , wherein the one or more protease inhibitors is aprotinin and/or soybean trypsin inhibitor.

8. The method of alleviating the symptoms of the inflammatory bowel disease according to claim 7 , wherein the GM-CSF comprises a conjugate that extends the half-life of the active ingredient.

9. The method of alleviating the symptoms of the inflammatory bowel disease according to claim 7 , wherein the conjugate that extends the half-life of the active ingredient is albumin or a fatty acid.

10. The method of alleviating the symptoms of the inflammatory bowel disease according to claim 2 , wherein said inflammatory bowel disease is Crohn's disease, and wherein the composition is for local administration into the lumen of an affected area of the intestines.

Assignments (2)
CHANGE OF NAME Recorded Sep 5, 2018
From: REPONEX PHARMACEUTICALS APS
To: REPONEX PHARMACEUTICALS A/S
Reel/Frame 047749/0257 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Oct 19, 2017
From: UTTENTHAL, LARS OTTO
To: REPONEX PHARMACEUTICALS APS
Reel/Frame 043904/0886 →
Priority Claims (1)
DK 2014 70461 · Jul 24, 2014 · national
Continuity (1)
Related Publication 20170196937A1 · Jul 13, 2017
Cited By (1)
US 12,698,306