IP Library › Granted Patent US 9,981,901
Granted Patent B2
US 9,981,901 · App. 15/356,292 · Granted May 29, 2018

IRE-1α inhibitors

Inventors: John B. Patterson (Ventura, CA); David G. Lonergan (San Marcos, CA); Gary A. Flynn (Tucson, AZ); Qingping Zeng (Thousand Oaks, CA); Peter V. Pallai (Carlsbad, CA)
Assignee: FOSUN ORINOVE PHARMATECH, INC.
C07C65/21A61K31/166C07C65/11C07C65/26C07C233/65C07C235/42
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Quick Facts
Patent No.
US 9,981,901
App. No.
15/356,292
Granted
May 29, 2018
Kind
B2
Abstract

Compounds which directly inhibit IRE-1α activity in vitro, prodrugs, and pharmaceutically acceptable salts thereof. Such compounds and prodrugs are useful for treating diseases associated with the unfolded protein response and can be used as single agents or in combination therapies.

Claims (3)

1. An IRE-1α inhibitor, wherein the IRE-1α inhibitor is:

or a pharmaceutically acceptable salt thereof.

2. A pharmaceutical composition comprising the IRE-1α inhibitor of claim 1 .

Assignments (3)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Mar 22, 2018
From: SHANGHAI FOSUN PHARMACEUTICAL INDUSTRIAL DEVELOPMENT CO. LTD.
To: FOSUN ORINOVE PHARMATECH, INC.
Reel/Frame 045320/0357 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded May 23, 2017
From: MANNKIND CORPORATION
To: SHANGHAI FOSUN PHARMACEUTICAL INDUSTRIAL DEVELOPMENT CO. LTD.
Reel/Frame 042483/0622 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Apr 24, 2017
From: PATTERSON, JOHN B.; LONERGAN, DAVID G.; FLYNN, GARY A.; ZENG, QINGPING; PALLAI, PETER V.
To: MANNKIND CORPORATION
Reel/Frame 042322/0623 →
Continuity (6)
Continuation 14969837 · Dec 15, 2015
Division 14078792 · Nov 13, 2013
Division 12941530 · Nov 8, 2010
Continuation 12135571 · Jun 9, 2008
Provisional Application 60942743 · Jun 8, 2007
Related Publication 20170152206A1 · Jun 1, 2017