IP Library › Granted Patent US 10,426,763
Granted Patent B2
US 10,426,763 · App. 15/356,766 · Granted Oct 1, 2019

Pharmaceutical compositions comprising glitazones and NRF2 activators

Inventor: Bjoern Colin Kahrs (Collonge-Bellerive, CH)
Assignee: Bjoern Colin Kahrs
A61K31/4439A61K9/0053A61K31/05A61K31/12A61K31/16A61K31/19A61K31/216A61K31/225A61K31/26A61K31/385A61K31/426A61K31/47Y02A50/395Y02A50/414
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Quick Facts
Patent No.
US 10,426,763
App. No.
15/356,766
Granted
Oct 1, 2019
Kind
B2
Abstract

The invention relates to pharmaceutical compositions comprising PPAR agonists and Nrf2 activators and methods of using combinations of PPAR agonists and Nrf2 activators for treating diseases such as psoriasis, asthma, multiple sclerosis, inflammatory bowel disease, and arthritis.

Claims (9)

1. A method of alleviating multiple sclerosis or a clinical symptom thereof or delaying the onset of multiple sclerosis or a clinical symptom thereof in a patient, comprising the co-administration of therapeutically effective amounts of an Nrf2 activator selected from the fumaric acid esters and salts thereof and a PPAR gamma agonist selected from glitazones and salt forms thereof to said patient.

2. The method according to claim 1 , wherein the glitazone is selected from the group of pioglitazone and its salt forms and rosiglitazone and its salt forms.

3. The method according to claim 1 , wherein the glitazone is pioglitazone.

4. The method according to claim 1 , wherein the glitazone is pioglitazone hydrochloride.

5. The method according to claim 1 , wherein the Nrf2 activator is selected from the group of monoalkyl fumarates and dialkyl fumarates.

6. The method according to claim 1 , wherein the Nrf2 activator is selected from the group of monomethyl fumarate, dimethyl fumarate, monoethyl fumarate and diethyl fumarate.

7. The method according to claim 1 , wherein the PPAR gamma agonist is rosiglitazone.

8. The method according to claim 1 , wherein the PPAR gamma agonist is rosiglitazone maleate.

9. The method according to claim 1 , wherein said co-administration is an oral administration.

Assignments (2)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Dec 21, 2017
From: KAHRS, BJOERN C.
To: ARES TRADING S.A.
Reel/Frame 044458/0264 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Dec 21, 2017
From: ARES TRADING S.A.
To: KAHRS, BJOERN COLIN
Reel/Frame 044458/0291 →
Priority Claims (2)
EP 11194292 · Dec 19, 2011 · regional
EP 12004652 · Jun 21, 2012 · regional
Continuity (4)
Continuation 14363042
Continuation In Part 13654632 · Oct 18, 2012
Provisional Application 61663761 · Jun 25, 2012
Related Publication 20170065571A1 · Mar 9, 2017
Cited By (3)
US 12,239,626 US 12,247,071 US 12,310,939