IP Library Granted Patent US 10,080,777
Granted Patent B2
US 10,080,777 · App. 15/375,523 · Granted Sep 25, 2018

Syndecan peptides and polypeptides and uses thereof

Inventor: Alan Rapraeger (Stoughton, WI)
Assignee: Wisconsin Alumni Research Foundation
A61K38/177
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Quick Facts
Patent No.
US 10,080,777
App. No.
15/375,523
Granted
Sep 25, 2018
Kind
B2
Abstract

The invention provides for peptides from syndecan 4 and methods of use therefor. These peptides can inhibit α6β4 integrin interaction with EGFR, thereby preventing tumor cell growth and tissue invasion, or inhibiting scarring and/or pathologic neovascularization.

Claims (11)

1. A method of inhibiting pathologic neovascularization or inhibiting scarring in a subject in need thereof, comprising administering to said subject a peptide segment consisting of between 45 and 100 amino acid residues and comprising about 45 residues of SEQ ID NO:1, including residues 87-131 of SEQ ID NO:1 (SEQ ID NO:4), whereby pathologic neovascularization or scarring is inhibited in the subject.

2. The method of claim 1 , wherein the peptide segment is 45, 46, 47, 48, 49, 50, 51, 52, 53, 54, 55, 60, 65, 70, 75, 80, 85, 90, 95 or 100 amino acid residues in length.

3. The method of claim 1 , wherein the peptide segment is between 45 and 54 amino acid residues in length, between 45 and 65 amino acid residues in length, or between 45 and 75 amino acid residues in length.

4. The method of claim 1 , wherein the peptide segment consists essentially of residues 87-131 of SEQ ID NO:1 (SEQ ID NO:4).

5. The method of claim 1 , wherein the peptide segment consists of residues 87-131 of SEQ ID NO:1 (SEQ ID NO:4).

6. The method of claim 1 , wherein the peptide segment consists essentially of residues 78-131 of SEQ ID NO:1 (SEQ ID NO:5).

7. The method of claim 1 , wherein said peptide segment consists of residues 78-131 of SEQ ID NO:1 (SEQ ID NO: 5).

8. The method of claim 1 , wherein the peptide segment comprises all D amino acid, all L amino acids, or a mixture of D and L amino acids.

9. The method of claim 1 , wherein pathologic neovascularization is inhibited in the subject.

10. The method of claim 9 , wherein said pathologic neovascularization involves activated vascular endothelial cells.

11. The method of claim 1 , wherein scarring is inhibited in the subject.

Assignments (2)
CONFIRMATORY LICENSE Recorded Jul 3, 2018
From: UNIVERSITY OF WISCONSIN MADISON
To: NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT
Reel/Frame 046473/0976 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Mar 14, 2017
From: RAPRAEGER, ALAN
To: WISCONSIN ALUMNI RESEARCH FOUNDATION
Reel/Frame 041568/0578 →
Continuity (5)
Continuation 14688703 · Apr 16, 2015
Division 13936872 · Jul 8, 2013
Provisional Application 61784930 · Mar 14, 2013
Provisional Application 61669551 · Jul 9, 2012
Related Publication 20170087210A1 · Mar 30, 2017