IP Library › Granted Patent US 10,471,145
Granted Patent B2
US 10,471,145 · App. 15/414,533 · Granted Nov 12, 2019

Methods for treating cancer using nanoparticle complexes of paclitaxel, rituximab, and albumin

Inventors: Svetomir N. Markovic (Rochester, MN); Wendy K. Nevala (Rochester, MN)
Assignee: Mayo Foundation for Medical Education and Research
A61K39/39558A61K9/0019A61K9/14A61K9/51A61K9/5169A61K31/282A61K31/337A61K31/555A61K33/24A61K39/395A61K41/0052A61K45/06A61K47/643A61K47/6801A61K47/6803A61K47/6845A61K47/6849A61K47/6851A61K47/6855A61K47/6863A61K47/6865A61K47/6867A61K47/6929A61K47/6931C07K16/22C07K16/2863C07K16/2887C07K16/2893C07K16/3015C07K16/32A61K2039/505A61K2039/545A61K2039/6056B82Y5/00C07K2317/21C07K2317/24C07K2317/73C07K2317/92C07K2317/94
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Quick Facts
Patent No.
US 10,471,145
App. No.
15/414,533
Granted
Nov 12, 2019
Kind
B2
Abstract

Described are stable nanoparticle complexes comprising paclitaxel, albumin and ofatumumab. The nanoparticle complexes are suitable for the treatment of cancer.

Claims (15)

1. A method for treating cancer in a subject in need thereof, the method comprising administering to the subject a therapeutically effective amount of a pharmaceutical composition comprising a pharmaceutically acceptable carrier and antibody-albumin nanoparticle complexes, said complexes comprising albumin, a rituximab antibody, and paclitaxel, wherein the nanoparticle complexes have been pre-formed in vitro by mixing aqueous albumin-paclitaxel nanoparticies with the antibody under conditions to form the nanoparticle complexes, such that the nanoparticle complexes have CD20 binding specificity, wherein the cancer expresses CMG, and wherein the average diameter of said complexes is between 0.1 μm and 1 μm.

2. The method of claim 1 , wherein the average diameter of said complexes is between 0.1 μm and 0.9 μm.

3. The method of claim 1 , wherein the average diameter of said complexes is between 0.1 μm and 0.3 μm.

4. The method of claim 1 , wherein the ratio of albumin-paclitaxel nanoparticle to antibody is between 5:1 and 1:2.5.

5. The method of claim 1 , wherein the pharmaceutical composition is administered by intravenous injection.

6. The method of claim 1 , wherein the subject is a human.

7. The method of claim 1 , wherein the cancer is leukemia or lymphoma.

8. The method of claim 1 , wherein the therapeutically effective amount is between about 30 mg/m 2 and about 70 mg/m 2 antibody.

9. The method of claim 1 , wherein the therapeutically effective amount is between about 5 mg/kg and about 20 mg/kg antibody.

10. The method of claim 1 , wherein the therapeutically effective amount is between about 50 mg/m 2 and about 175 mg/m 2 albumin-paclitaxel nanoparticles.

11. The method of claim 1 , wherein the pharmaceutical composition is administered from about once a month to about three times a month.

12. The method of claim 1 , wherein the pharmaceutical composition is administered three times per 28 day cycle for at least two cycles.

13. The method of claim 1 , wherein said composition comprises an alkylating agent.

14. The method of claim 13 , wherein said alkylating agent is a platinum compound.

15. The method of claim 1 , wherein the pharmaceutically acceptable carrier is saline, water, lactic acid, mannitol, or a combination thereof.

Assignments (1)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jan 26, 2017
From: MARKOVIC, SVETOMIR N.; NEVALA, WENDY K.
To: MAYO FOUNDATION FOR MEDICAL EDUCATION AND RESEARCH
Reel/Frame 041098/0372 →
Continuity (5)
Continuation 15202115 · Jul 5, 2016
Continuation 14432979
Provisional Application 61708575 · Oct 1, 2012
Provisional Application 61725293 · Nov 12, 2012
Related Publication 20170128588A1 · May 11, 2017
Cited By (2)
US 12,364,754 US 12,403,119