IP Library Granted Patent US 10,251,887
Granted Patent B2
US 10,251,887 · App. 15/438,244 · Granted Apr 9, 2019

Methods and compositions to reduce oxidative stress

Inventor: Louis M. Messina (Westborough, MA)
Assignee: University of Massachusetts
A61K31/519A61K31/198A61K31/375A61K45/06A61K48/005A61K31/495A61K35/13A61K2300/00C12N2799/022C12P13/10
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Quick Facts
Patent No.
US 10,251,887
App. No.
15/438,244
Granted
Apr 9, 2019
Kind
B2
Abstract

The invention relates to therapeutic applications for compositions that reduce the level of oxidative stress on cells in vivo or in vitro. The invention describes methods for improving the therapeutic properties of stem cells. The invention also provides combination therapies that are useful to balance the oxidative microenvironment of cells in vivo or in vitro.

Claims (25)

1. A method of treating atherosclerosis in a subject, the method comprising identifying a subject who has atherosclerosis and administering to the subject active agents consisting of:

a. L-arginine,

b. tetrahydrobiopterin, sepiapterin, or dihydrobiopterin, or any combination thereof, and

c. ascorbic acid or ascorbate;

wherein the ratio of (a):(b) is 1-30:1; and

wherein the ratio of (b):(c) is 1:0.1-15.

2. The method of claim 1 , comprising administering:

a. L-arginine;

b. tetrahydrobiopterin; and

c. ascorbic acid or ascorbate.

3. The method of claim 1 , comprising administering:

88.5 mg/kg/day L-arginine;

10 mg/kg/day tetrahydrobiopterin; and

88.5 mg/kg/day ascorbic acid or ascorbate.

4. The method of claim 1 , wherein the method comprises administering to the subject a pharmaceutical composition, wherein the active ingredients of the composition consist of:

a. L-arginine,

b. tetrahydrobiopterin, sepiapterin, or dihydrobiopterin, or any combination thereof, and

c. ascorbic acid or ascorbate;

wherein the ratio of (a):(b) is 1-30:1; and

wherein the ratio of (b):(c) is 1:0.1-15.

5. The method of claim 4 , wherein the pharmaceutical composition is formulated as tablets, capsules, powders, granules, or solutions for oral ingestion.

6. The method of claim 4 , wherein the pharmaceutical composition comprises one or more excipients selected from the group consisting of:

hydroxypropyl methylcellulose; sodium carboxymethyl cellulose; and

polyvinylpyrrolidine.

7. The method of claim 1 , wherein the treatment reduces vascular plaque formation.

Assignments (2)
CONFIRMATORY LICENSE Recorded Oct 30, 2017
From: UNIVERSITY OF MASSACHUSETTS MEDICAL SCH
To: NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT
Reel/Frame 044318/0434 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Apr 25, 2017
From: MESSINA, LOUIS M.
To: UNIVERSITY OF MASSACHUSETTS
Reel/Frame 042134/0896 →
Continuity (5)
Division 14535690 · Nov 7, 2014
Division 13386462
Provisional Application 61357179 · Jun 22, 2010
Provisional Application 61227768 · Jul 22, 2009
Related Publication 20170258796A1 · Sep 14, 2017