IP Library Granted Patent US 10,080,726
Granted Patent B2
US 10,080,726 · App. 15/505,414 · Granted Sep 25, 2018

Method for treating hyperhidrosis with dexmecamylamine

Inventor: Merouane Bencherif (Winston-Salem, NC)
A61K31/13A61K9/0053A61K9/20
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Quick Facts
Patent No.
US 10,080,726
App. No.
15/505,414
Granted
Sep 25, 2018
Kind
B2
Abstract

The present invention relates to dexmecamylamine and the use of dexmecamylamine, substantially free of exo-R-mecamylamine, in the treatment of hyperhidrosis.

Claims (19)

1. A method of treating hyperhidrosis, the method comprising the administration of a therapeutically effective amount of dexmecamylamine or a pharmaceutically acceptable salt thereof, substantially free of exo-R-mecamylamine, to a subject with hyperhidrosis, wherein the dexmecamylamine or a pharmaceutically acceptable salt thereof is administered in an amount from about 0.1 mg to about 4.0 mg.

2. A method of treating hyperhidrosis, the method comprising the oral administration of dexmecamylamine or a pharmaceutically acceptable salt thereof in an amount from about 0.1 mg to about 2.0 mg once daily, substantially free of exo-R-mecamylamine, to a subject with hyperhidrosis.

3. The method according to claim 2 , wherein the dexmecamylamine or a pharmaceutically acceptable salt thereof is orally administered in an amount of about 0.2 mg once daily.

4. The method according to claim 2 , wherein the dexmecamylamine or a pharmaceutically acceptable salt thereof is orally administered in an amount of about 0.5 mg once daily.

5. The method according to claim 2 , wherein the dexmecamylamine or a pharmaceutically acceptable salt thereof is orally administered in an amount of about 1.0 mg once daily.

6. The method according to claim 2 , wherein the dexmecamylamine or a pharmaceutically acceptable salt thereof is orally administered in an amount of about 2.0 mg once daily.

7. The method according to claim 2 , wherein the dexmecamylamine or a pharmaceutically acceptable salt thereof is orally administered in tablet form.

8. A method of treating hyperhidrosis comprising the oral administration of dexmecamylamine or a pharmaceutically acceptable salt thereof in an amount from about 0.1 mg to about 2.0 mg once daily, substantially free of exo-R-mecamylamine, to a subject with hyperhidrosis, wherein the administration of dexmecamylamine is sufficient to affect sweating in a patient in at least one location with an Hyperhidrosis Disease Severity Scale change of >1.

9. The method according to claim 8 , wherein the administration of dexmecamylamine is sufficient to affect sweating in a patient in at least two locations with an HDSS change of >0.5, in each location.

10. The method according to claim 8 , wherein the location is selected from axillary, palmoplantar, face/scalp, or generalized.

11. The method according to claim 2 , wherein the hyperhidrosis is primary hyperhidrosis.

12. The method according to claim 2 , wherein the subject is a human.

13. The method according to claim 1 , wherein the dexmecamylamine or a pharmaceutically acceptable salt thereof is administered once daily.

14. The method according to claim 1 , wherein the dexmecamylamine or a pharmaceutically acceptable salt thereof is administered more than once daily.

15. The method according to claim 1 , wherein the dexmecamylamine or a pharmaceutically acceptable salt thereof is orally administered in an amount of about 1.0 mg.

16. The method according to claim 1 , wherein the dexmecamylamine or a pharmaceutically acceptable salt thereof is orally administered in an amount of about 2.0 mg.

17. The method according to claim 1 , wherein the dexmecamylamine or a pharmaceutically acceptable salt thereof is orally administered in an amount of about 4.0 mg.

18. The method according to claim 1 , wherein the hyperhidrosis is primary hyperhidrosis.

19. The method according to claim 1 , wherein the dexmecamylamine or a pharmaceutically acceptable salt thereof is orally administered in tablet form.

Assignments (3)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Sep 20, 2018
From: CATALYST BIOSCIENCES, INC.
To: ATACAMA THERAPEUTICS, INC.
Reel/Frame 046931/0325 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Sep 20, 2018
From: BENCHERIF, MEROUANE
To: TARGACEPT, INC.
Reel/Frame 047118/0761 →
CHANGE OF NAME Recorded Sep 20, 2018
From: TARGACEPT, INC.
To: CATALYST BIOSCIENCES, INC.
Reel/Frame 047118/0810 →
Continuity (2)
Provisional Application 62040477 · Aug 22, 2014
Related Publication 20170266132A1 · Sep 21, 2017