IP Library › Granted Patent US 10,682,424
Granted Patent B2
US 10,682,424 · App. 15/561,547 · Granted Jun 16, 2020

Compositions and method for reducing seizures

Inventors: Gordon Fishell (Larchmont, NY); Jordane Dimidschstein (Seraing, BE)
Assignee: New York University
A61K48/0066A61K38/1796C07K14/705C07K14/723C12N7/00C12N15/86A61K38/00C12N2750/14121C12N2750/14143C12N2830/008C12N2830/30C12N2830/42C12N2830/48C12N2830/50
View Patent ↗
Loading inventors, assignments & file history…
Monitor This Case
Get email alerts when status or documents change.
Order Certified Copies
Most orders are placed with the USPTO same day — all within 24 business hours.
Order via The Patent Place →
Pre-filled with this patent's details
Quick Facts
Patent No.
US 10,682,424
App. No.
15/561,547
Granted
Jun 16, 2020
Kind
B2
Abstract

Provided are compositions and methods for prophylaxis and/or therapy of disorders that involve seizures. The compositions and methods relate to a recombinant adeno-associated virus (rAAV) comprising a I56i enhancer sequence, and a sequence encoding hM3Dq modified muscarinic receptor (Gq-DREADD). The method includes introducing the rAAV into interneurons of an individual such that Gq-DREADD is expressed in interneurons of the individual. The method can further comprise administering to the individual an agonist of the Gq-DREADD, such for reducing or preventing seizures.

Claims (5)

1. A method for prophylaxis and/or therapy for seizures in an individual mammal in need thereof, the method comprising administering with a stereotactic injection into the somatosensory cortex, hippocampus and/or striatum of the mammal's brain a recombinant adeno-associated virus (rAAV) comprising a sequence encoding a I56i enhancer and a sequence encoding hM3Dq modified muscarinic receptor (Gq-DREADD) such that neurons of brain of the individual mammal comprise the I56i enhancer sequence that is operably linked to the sequence encoding the Gq-DREADD, wherein the Gq-DREADD is only expressed in adult GABA-ergic interneurons, and subsequently administering to the individual an effective amount of clozapine-N4-oxide (CNO), wherein one or more seizures are inhibited or prevented.

2. The method of claim 1 , wherein the individual is experiencing a seizure at time of the administering the CNO and wherein the severity of the seizure is reduced subsequent to the administering.

3. The method of claim 1 , wherein the seizure is selected from a partial seizure or a generalized seizure.

4. The method of claim 1 , wherein the individual mammal has, is suspected of having, or has been diagnosed with epilepsy.

5. The method of claim 1 , wherein the individual mammal has been diagnosed with pharmaco-resistant epilepsy.

Assignments (1)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jan 17, 2019
From: FISHELL, GORDON; DIMIDSCHSTEIN, JORDANE
To: NEW YORK UNIVERSITY
Reel/Frame 048043/0251 →
Continuity (2)
Provisional Application 62140631 · Mar 31, 2015
Related Publication 20180078658A1 · Mar 22, 2018