IP Library › Granted Patent US 10,603,334
Granted Patent B2
US 10,603,334 · App. 15/570,210 · Granted Mar 31, 2020

Targeting NAD

Inventors: Lindsay Edward Wu (Waterloo, AU); David A. Sinclair (Chestnut Hill, MA)
Assignee: NewSouth Innovation Pty. Limited
A61K31/706A61K31/443A61K31/455A61K31/52A61K31/7076A61K38/45A61P25/02C12Y204/02012C12Y207/07001
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Quick Facts
Patent No.
US 10,603,334
App. No.
15/570,210
Granted
Mar 31, 2020
Kind
B2
Abstract

Methods and compositions for preventing or treating peripheral neuropathy, cognitive deficits, inactivity, depression, chemotherapy and/or radiotherapy induced peripheral neuropathy and cognitive deficits, and improving cognitive performance, in a subject in need thereof are disclosed. The disclosed methods include the step of administering to the subject an effective amount of an agent that increases the level of NAD + in the subject.

Claims (15)

1. A method for prophylactically treating chemotherapy induced cognitive impairments (CICI) in a subject, comprising administering to a subject who has undergone exposure to a chemotherapy agent, is undergoing exposure to a chemotherapy agent, or will undergo exposure to a chemotherapy agent, an effective amount of an agent that increases the level of NAD + in the subject, whereby chemotherapy agent-induced cognitive impairments (CICI) are prophylactically treated,

wherein the agent that increases the level of NAD + is an NAD + precursor selected from nicotinamide mononucleotide (NMN), nicotinic acid, nicotinamide, nicotinamide riboside (NR), nicotinic acid mononucleotide, nicotinic acid riboside, 5-aminoimidazole-4-carboxamide ribonucleotide (AICAR), adenosine, adenine, and adenosine monophosphate.

2. The method of claim 1 , wherein the chemotherapy agent induced neurotoxic damage prophylactically treated comprises chemotherapy induced peripheral neuropathies (CIPN).

3. The method of claim 1 , wherein the chemotherapy agent induced neurotoxic damage prophylactically treated comprises chemotherapy induced inactivity.

4. The method of claim 1 , wherein the chemotherapy agent induced neurotoxic damage prophylactically treated comprises chemotherapy induced depression, anxiety, melancholy, post-traumatic stress disorder, impaired sleep, circadian rhythm disorders, or other mental health/psychological disorder.

5. The method of claim 1 , wherein the agent that increases the level of NAD+ in the subject is administered at the same time as the subject undergoes exposure to the chemotherapy agent.

6. The method of claim 1 , wherein the neurotoxic damage prophylactically treated comprises pain and/or peripheral neuropathy.

7. The method of claim 1 , wherein the neurotoxic damage prophylactically treated comprises inactivity, lethargy, or malaise.

8. The method of claim 1 , wherein the neurotoxic damage prophylactically treated comprises depression, anxiety, melancholy, post-traumatic stress disorder or other mental health/psychological disorder.

9. The method of claim 1 , wherein the chemotherapy agent is selected from cisplatin, carboplatin, oxaliplatin, cyclophosphamide, altretamine, plicamydin, chlorambucil, chlormethine, ifosfamide, melphalan, carmustine, fotemustine, lomustine, streptozocin, busulfan, dacarbazine, mechlorethamine, procarbazine, temozolomide, thioTEPA, uramustine, paclitaxel, docetaxel, vinblastine, vincristine, vindesine, vinorelbine, hexamethylmelamine, etoposide, teniposide, methotrexate, pemetrexed, raltitrexed, cladribine, clofarabine, fludarabine, mercaptopurine, tioguanine, capecitabine, cytarabine, fluorouracil, fluxuridine, gemcitabine, daunorubicin, doxorubicin, epirubicin, idarubicin, mitoxantrone, valrubicin, bleomycin, hydroxyurea, mitomycin, topotecan, irinotecan, aminolevulinic acid, methyl aminolevulinate, porfimer sodium, verteporfin, alitretinoin, altretamine, amsacrine, anagrelide, arsenic trioxide, asparaginase, bexarotene, bortezomib, celecoxib, denileukin, diftitox, erlotinib, estramustine, gefitinib, hydroxycarbamide, imatinib, pentostatin, masoprocol, mitotane, pegaspargase, and tretinoin, or combinations thereof.

10. The method of claim 1 , wherein the agent that increases the level of NAD + is an activator to an enzyme involved in NAD + biosynthesis.

11. The method of claim 1 , wherein the agent that increases the level of NAD + is administered at a dose of between 0.5-5 grams per day.

12. The method of claim 1 , wherein the subject is a human.

13. The method of claim 1 , comprising administering the agent that increases the level of NAD+ in the subject before the subject undergoes exposure to the chemotherapy agent.

14. The method of claim 1 , comprising administering the agent that increases the level of NAD+ in the subject after the subject undergoes exposure to the chemotherapy agent.

Assignments (3)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Mar 7, 2024
From: NEWSOUTH INNOVATIONS PTY LTD
To: METRO BIOTECH NSW PTY LTD
Reel/Frame 066685/0624 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Mar 7, 2024
From: METRO BIOTECH NSW PTY LTD
To: METRO INTERNATIONAL BIOTECH, LLC
Reel/Frame 066685/0660 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Dec 20, 2017
From: WU, LINDSAY EDWARD; SINCLAIR, DAVID A.
To: NEWSOUTH INNOVATIONS PTY. LIMITED
Reel/Frame 044447/0180 →
Continuity (2)
Provisional Application 62153876 · Apr 28, 2015
Related Publication 20180125871A1 · May 10, 2018
Cited By (2)
US 12,344,629 US 12,358,940