IP Library Granted Patent US 10,512,635
Granted Patent B2
US 10,512,635 · App. 15/580,850 · Granted Dec 24, 2019

Uses of benzimidazole derivative for nocturnal acid breakthrough

Inventors: Ha Jin Lee (Seoul, KR); Bong Tae Kim (Gyeonggi-do, KR); Hyun Kim (Gyeonggi-do, KR); Ji Yeon Nam (Seoul, KR); Jie Eun Park (Gyeonggi-do, KR); Geun Seog Song (Seoul, KR); Shin Young Ryu (Gyeonggi-do, KR); Shinichi Koizumi (Aichi, JP); Nobuyuki Takahashi (Aichi, JP); Masaomi Tajimi (Aichi, JP)
Assignees: CJ Healthcare Corporation; RaQualia Pharma Inc.
A61K31/4184A61K9/20A61K9/28A61P1/04
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Quick Facts
Patent No.
US 10,512,635
App. No.
15/580,850
Granted
Dec 24, 2019
Kind
B2
Abstract

The present invention relates to a use of benzimidazole derivative compounds for improvement and treatment of nocturnal acid breakthrough (NAB). The benzimidazole derivative compounds can mere effectively prevent and treat gastric acid-related diseases by effectively improving and treating nocturnal nocturnal acid breakthrough symptoms.

Claims (13)

1. A method for treating nocturnal acid breakthrough, comprising administering a pharmaceutical composition to a subject in need thereof, wherein the composition comprises a compound represented by Chemical Formula 1 or a pharmaceutically acceptable salt thereof, as an active ingredient,

2. The method of claim 1 , wherein the composition comprises 10 mg to 500 mg of the compound represented by Chemical Formula 1 or the pharmaceutically acceptable salt thereof.

3. A method for treating nocturnal acid breakthrough, comprising administering a unit dosage form to a subject in need thereof, wherein the unit dosage form comprises 10 mg to 500 mg of a compound represented by Chemical Formula 1 or a pharmaceutically acceptable salt thereof,

4. The method of claim 3 , wherein the unit dosage form further comprises a pharmaceutically acceptable carrier.

5. The method of claim 3 , wherein the subject is a patient suffering from a disease selected from the group consisting of erosive gastroesophageal reflux disease (GERD), non-erosive gastroesophageal reflux disease (NERD), gastric ulcer, Barrett's esophagus, and esophagus motility disorder.

6. The method of claim 3 , wherein the unit dosage form alleviates or ameliorates symptoms of heartburn.

7. The method of claim 3 , wherein the unit dosage form is administered before dinner or bedtime.

8. The method of claim 3 , wherein the unit dosage form is administered one to three times a day to a lowest acceptable daily dose.

9. The method of claim 3 , wherein the unit dosage form is a unit dosage form for oral administration.

10. The method of claim 3 , wherein the percentage of time when gastric pH is maintained at 4 or higher out of 12 hours after the administration of the unit dosage form is 65% or more.

11. The method of claim 3 , wherein the gastric pH reaches 4 within 2 hours after the administration of the unit dosage form.

12. The method of claim 1 , wherein the composition comprises 50 mg to 200 mg of the compound represented by Chemical Formula 1 or the pharmaceutically acceptable salt thereof.

13. The method of claim 3 , wherein the unit dosage form comprises 50 mg to 200 mg of the compound represented by Chemical Formula 1 or the pharmaceutically acceptable salt thereof.

Assignments (3)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Apr 27, 2021
From: RAQUALIA PHARMA INC.
To: HK INNO.N CORPORATION
Reel/Frame 056052/0108 →
CHANGE OF NAME Recorded Aug 12, 2020
From: CJ HEALTHCARE CORPORATION
To: HK INNO.N CORPORATION
Reel/Frame 053469/0285 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Dec 8, 2017
From: LEE, HA JIN; KIM, BONG TAE; KIM, HYUN; NAM, JI YEON; PARK, JIE EUN; SONG, GEUN SEOG; RYU, SHIN YOUNG; KOIZUMI, SHINICHI; TAKAHASHI, NOBUYUKI; TAJIMI, MASAOMI
To: CJ HEALTHCARE CORPORATION; RAQUALIA PHARMA INC.
Reel/Frame 044339/0635 →
Continuity (2)
Provisional Application 62172680 · Jun 8, 2015
Related Publication 20180338954A1 · Nov 29, 2018